共 50 条
- [31] Preclinical characterization of PRT3789, a potent and selective SMARCA2 targeted degraderCANCER RESEARCH, 2022, 82 (12)Hulse, Michael论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAAgarwal, Anjana论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAWang, Min论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USACarter, Jack论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USASivakumar, Monisha论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAVidal, Brian论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USABrown, Justin论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAMoore, Andrew论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAGrego, Alexander论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USABhagwat, Neha论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USARager, Joseph论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USALu, Liang论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USABasch, Corey论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USABersch, Klare论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USADai, Chaofeng论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAPitis, Philip论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USACombs, Andrew论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USARuggeri, Bruce论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAVaddi, Kris论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAScherle, Peggy论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USAIto, Koichi论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut, Wilmington, DE USA Prelude Therapeut, Wilmington, DE USA
- [32] Discovery and characterization of potent, selective CBP degradersCANCER RESEARCH, 2023, 83 (07)La Bonte, Laura论文数: 0 引用数: 0 h-index: 0Sappal, Darshan论文数: 0 引用数: 0 h-index: 0
- [33] Discovery of highly potent, selective and efficacious STAT3 PROTAC degraders capable of achieving long-lasting tumor regressionCANCER RESEARCH, 2024, 84 (06)Zhou, Haibin论文数: 0 引用数: 0 h-index: 0Wu, Dimin论文数: 0 引用数: 0 h-index: 0Bai, Longchuan论文数: 0 引用数: 0 h-index: 0Acharyya, Ranjan K.论文数: 0 引用数: 0 h-index: 0Metwally, Hoda论文数: 0 引用数: 0 h-index: 0McEachern, Donna论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [34] SMARCA2 (BRM) degraders promotes differentiation and inhibit proliferation in AML modelsCANCER RESEARCH, 2023, 83 (07)Agarwal, Anjana论文数: 0 引用数: 0 h-index: 0Osinubi, Olusola Peace论文数: 0 引用数: 0 h-index: 0Vykuntam, Komali论文数: 0 引用数: 0 h-index: 0Fultang, Norman论文数: 0 引用数: 0 h-index: 0Bhagwat, Neha论文数: 0 引用数: 0 h-index: 0Heiser, Diane论文数: 0 引用数: 0 h-index: 0Vaddi, Kris论文数: 0 引用数: 0 h-index: 0Ito, Koichi论文数: 0 引用数: 0 h-index: 0Scherle, Peggy论文数: 0 引用数: 0 h-index: 0
- [35] Discovery of PRT3789, a first-in-class potent and selective SMARCA2 degrader in clinical trials for the treatment of patients with SMARCA4 mutated cancersMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Ito, Koichi论文数: 0 引用数: 0 h-index: 0Hulse, Michael论文数: 0 引用数: 0 h-index: 0Agarwal, Anjana论文数: 0 引用数: 0 h-index: 0Carter, Jack论文数: 0 引用数: 0 h-index: 0Sivakumar, Monisha论文数: 0 引用数: 0 h-index: 0Vykuntam, Komali论文数: 0 引用数: 0 h-index: 0Wang, Min论文数: 0 引用数: 0 h-index: 0Cowart, Miles论文数: 0 引用数: 0 h-index: 0Cote, Joy论文数: 0 引用数: 0 h-index: 0-MacDonald, William Gowen论文数: 0 引用数: 0 h-index: 0Torres, Brian Vidal论文数: 0 引用数: 0 h-index: 0Kurian, Justin论文数: 0 引用数: 0 h-index: 0Bhagwat, Neha论文数: 0 引用数: 0 h-index: 0Fultang, Norman论文数: 0 引用数: 0 h-index: 0Grego, Alexander论文数: 0 引用数: 0 h-index: 0Moore, Andrew论文数: 0 引用数: 0 h-index: 0Schwab, Ashley论文数: 0 引用数: 0 h-index: 0Burtell, Jessica论文数: 0 引用数: 0 h-index: 0Osinubi, Olusola Peace论文数: 0 引用数: 0 h-index: 0Spruance, Jacob论文数: 0 引用数: 0 h-index: 0Lu, Liang论文数: 0 引用数: 0 h-index: 0Pitis, Philip论文数: 0 引用数: 0 h-index: 0Basch, Corey论文数: 0 引用数: 0 h-index: 0Bersch, Klare论文数: 0 引用数: 0 h-index: 0Dai, Chaofeng论文数: 0 引用数: 0 h-index: 0Leal, Raul论文数: 0 引用数: 0 h-index: 0Shvartsbart, Artem论文数: 0 引用数: 0 h-index: 0Cao, Ganfeng论文数: 0 引用数: 0 h-index: 0Shen, Bo论文数: 0 引用数: 0 h-index: 0Wen, Patrick论文数: 0 引用数: 0 h-index: 0Rager, Joseph论文数: 0 引用数: 0 h-index: 0Kuskovsky, Ross论文数: 0 引用数: 0 h-index: 0Landman, Bob论文数: 0 引用数: 0 h-index: 0Emm, Tom论文数: 0 引用数: 0 h-index: 0Ruepp, Stefan论文数: 0 引用数: 0 h-index: 0Qin, Chunhua论文数: 0 引用数: 0 h-index: 0Paris, Gina论文数: 0 引用数: 0 h-index: 0Xavier, Jennifer论文数: 0 引用数: 0 h-index: 0Chiaverelli, Rachel论文数: 0 引用数: 0 h-index: 0Lee, Sang Hyun论文数: 0 引用数: 0 h-index: 0Geeganage, Sandy论文数: 0 引用数: 0 h-index: 0Lin, Hong论文数: 0 引用数: 0 h-index: 0Heiser, Diane论文数: 0 引用数: 0 h-index: 0Ruggeri, Bruce论文数: 0 引用数: 0 h-index: 0Babbar, Naveen论文数: 0 引用数: 0 h-index: 0Combs, Andrew论文数: 0 引用数: 0 h-index: 0Scherle, Peggy论文数: 0 引用数: 0 h-index: 0
- [36] Discovery of Highly Potent, Selective, and Efficacious Small Molecule Inhibitors of ERK1/2JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (04) : 1976 - 1991Ren, Li论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMoreno, David论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USABlake, James F.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGaudino, John J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGarrey, Rustam论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMetcalf, Andrew T.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USABurkard, Michael论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USARasor, Kevin论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAChen, Huifen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USADean, Brian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAGould, Stephen E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAPacheco, Patricia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAShahidi-Latham, Sheerin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAYin, Jianping论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAWest, Kristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAMoffat, John G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USASchwarz, Jacob B.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA
- [37] Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor AntagonistACS MEDICINAL CHEMISTRY LETTERS, 2011, 2 (03): : 213 - 218Eastwood, Paul论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainEsteve, Cristina论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainGonzalez, Jacob论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainFonquerna, Silvia论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainAiguade, Josep论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainCarranco, Ines论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainDomenech, Teresa论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainAparici, Monica论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainMiralpeix, Montserrat论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainAlberti, Joan论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainCordoba, Monica论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainFernandez, Raquel论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainPont, Merce论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainGodessart, Nuria论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainPrats, Neus论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainIsabel Loza, Maria论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago Compostela, Fac Pharm, Discovery Grp BioFarma, Santiago De Compostela 15782, Spain Almirall, R&D Ctr, Barcelona 08980, SpainIsabel Cadavid, Maria论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago Compostela, Fac Pharm, Discovery Grp BioFarma, Santiago De Compostela 15782, Spain Almirall, R&D Ctr, Barcelona 08980, SpainNueda, Arsenio论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, SpainVidal, Bernat论文数: 0 引用数: 0 h-index: 0机构: Almirall, R&D Ctr, Barcelona 08980, Spain Almirall, R&D Ctr, Barcelona 08980, Spain
- [38] Discovery of a highly potent and in vivo efficacious Bcl-xL selective inhibitorABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245Tao, Zhi-Fu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAWang, Le论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USANimmer, Paul M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USABoghaert, Erwin R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAChen, Jun论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAHasvold, Lisa A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAJin, Sha论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAKovar, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAMitten, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAOleksijew, Anatol论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAPark, Chang H.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAPetros, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAPhillips, Darren C.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USASmith, Morey论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USATahir, Stephen X.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USATse, Chris论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAWang, Xilu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAXiao, Yu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAZhang, Haichao论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USADeshayes, Kurt论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAFairbrother, Wayne J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAFlygare, John A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAHymowitz, Sarah G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAKoehler, Michael论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USANdubaku, Chudi论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USARawson, Tom论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAZobel, Kerry论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAColman, Peter M.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USACzabotar, Peter E.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAHuang, David C. S.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USALessene, Guillaume论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USASleebs, Brad E.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAWatson, Keith G.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Melbourne, Dept Med Biol, Melbourne, Vic, Australia Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USALeverson, Joel D.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USAElmore, Steven W.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USASouers, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs AbbVie, Canc Res, Abbott Pk, IL 60064 USA
- [39] Discovery of selective BRM ( SMARCA2) ATPase inhibitors for the treatment of BRG1 (SMARCA4) mutant cancersCANCER RESEARCH, 2024, 84 (06)Lee, Janice Y.论文数: 0 引用数: 0 h-index: 0Brooks, Nathan论文数: 0 引用数: 0 h-index: 0Antonakos, Brandon论文数: 0 引用数: 0 h-index: 0Perria, Bryan论文数: 0 引用数: 0 h-index: 0Langan, Candace论文数: 0 引用数: 0 h-index: 0Jones, Bonita D.论文数: 0 引用数: 0 h-index: 0Flack, Robert Stephen论文数: 0 引用数: 0 h-index: 0Li, Zhifang论文数: 0 引用数: 0 h-index: 0Terry, David论文数: 0 引用数: 0 h-index: 0Wallace, Ross论文数: 0 引用数: 0 h-index: 0Bondi, Robert论文数: 0 引用数: 0 h-index: 0Sis, Gereint论文数: 0 引用数: 0 h-index: 0Baracani, Ronee论文数: 0 引用数: 0 h-index: 0McVean, Maralee论文数: 0 引用数: 0 h-index: 0Kolakowski, Gabrielle论文数: 0 引用数: 0 h-index: 0Osimboni, Dayo论文数: 0 引用数: 0 h-index: 0Wilson, Kevin论文数: 0 引用数: 0 h-index: 0
- [40] Identification of a potent, orally-available SMARCA2/4 inhibitor with in vitro and in vivo activity in preclinical models of SMARCA4-mutant NSCLCCANCER RESEARCH, 2020, 80 (16)Drew, Allison E.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAJacques, Suzanne L.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAEichinger, Lindsey W.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAPantano, Chloe论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAMotwani, Vinny论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USATang, Cuyue论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAFarrow, Neil论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USABrach, Dorothy论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAHowe, Selene论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USARaimondi, Alejandra论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USADransfield, Daniel T.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USADuncan, Kenneth W.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAStickland, Kim论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USALampe, John论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USA