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- [21] Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitorBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (20) : 6188 - 6194Liddle, John论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandAtkinson, Francis L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandBarker, Michael D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandCarter, Paul S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandCurtis, Neil R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandDavis, Rob P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandDouault, Clement论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandDickson, Marion C.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandElwes, Dorothy论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandGarton, Neil S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandGray, Matthew论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandHayhow, Thomas G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandHobbs, Clare I.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandJones, Emma论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandLeach, Stuart论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandLeavens, Karen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandLewis, Huw D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandMcCleary, Scott论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandNeu, Margarete论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandPatel, Vipulkumar K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandPreston, Alex G. S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandRamirez-Molina, Cesar论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandShipley, Tracy J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandSkone, Philip A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandSmithers, Nick论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandSomers, Donald O.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandWalker, Ann L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandWatson, Robert J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, EnglandWeingarten, Gordon G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England GlaxoSmithKline R&D, Med Res Ctr, Stevenage, Herts, England
- [22] Discovery of SMD-3040 as a Potent and Selective SMARCA2 PROTAC Degrader with Strong in vivo Antitumor ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (15) : 10761 - 10781Yang, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USATu, Wenbin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAMiao, Bukeyan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAKaneshige, Atsunori论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAJiang, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USALeng, Lingying论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Meilin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
- [23] Discovery of highly potent, selective and efficacious STAT3 PROTAC degraders capable of achieving complete tumor regressionCANCER RESEARCH, 2024, 84 (06)Zhou, Haibin论文数: 0 引用数: 0 h-index: 0Wu, Dimin论文数: 0 引用数: 0 h-index: 0Bai, Longchuan论文数: 0 引用数: 0 h-index: 0Acharyya, Ranjan K.论文数: 0 引用数: 0 h-index: 0Metwally, Hoda论文数: 0 引用数: 0 h-index: 0McEachern, Donna论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [24] Combination therapy with selective SMARCA2 (BRM) degraders for treatment of SMARCA4 (BRG1)-deficient cancersCANCER RESEARCH, 2023, 83 (07)Hulse, Michael论文数: 0 引用数: 0 h-index: 0Elkins, Margot论文数: 0 引用数: 0 h-index: 0Burtell, Jessica论文数: 0 引用数: 0 h-index: 0Vykuntam, Komali论文数: 0 引用数: 0 h-index: 0Vaddi, Kris论文数: 0 引用数: 0 h-index: 0Combs, Andrew论文数: 0 引用数: 0 h-index: 0Ito, Koichi论文数: 0 引用数: 0 h-index: 0Scherle, Peggy论文数: 0 引用数: 0 h-index: 0
- [25] Development of novel, selective SMARCA2 (BRM) degraders for treatment of SMARCA4 (BRG1) mutated tumorsCANCER RESEARCH, 2020, 80 (16)Mazan, Andrzej论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandWrobel, Anna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandDreas, Agnieszka论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandRadzimierski, Adam论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandMichalik, Kinga论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandKowal, Anna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandWiklik, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandWnuk-Lipinska, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandNiedziejko, Paulina论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandKozlowska, Kamila论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandLosko, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandSzczesniak, Joanna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandSroka-Porada, Agnieszka论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandMartyka, Justyna论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandKulesza, Urszula论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandZuchowicz, Karol论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandZastawna, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandAlvarez, Jose论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandStasi, Luigi论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandLittlewood, Peter论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandRzymski, Tomasz论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, PolandBrzozka, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Ryvu Therapeut SA, Krakow, Poland Ryvu Therapeut SA, Krakow, Poland
- [26] GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (16) : 11177 - 11186Taylor, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USABailey, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USABelmont, Lisa D.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACampbell, Robert论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACantone, Nico论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACote, Alexandre论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACrawford, Terry D.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USACummings, Richard论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USADeMent, Kevin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USADuplessis, Martin论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAFlynn, Megan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAGood, Andrew C.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAHuang, Hon-Ren论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAJoshi, Shivangi论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USALeblanc, Yves论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAMurray, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USANasveschuk, Christopher G.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USANeiss, Adrianne论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAPoy, Florence论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USARomero, F. Anthony论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USASandy, Peter论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USATang, Yong论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USATsui, Vickie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAZawadzke, Laura论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USASims, Robert J., III论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAAudia, James E.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Flare Therapeut, 215 First St,Suite 150, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USAMagnuson, Steven R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USAAlbrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Constellation, Cambridge, MA 02142 USA Constellation, Cambridge, MA 02142 USACochran, Andrea G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Constellation, Cambridge, MA 02142 USA
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