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- [11] Discovery of YS-363 as a highly potent, selective, and orally efficacious EGFR inhibitorBIOMEDICINE & PHARMACOTHERAPY, 2023, 167He, Pengxing论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaJing, Jing论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaDu, Linna论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaZhang, Xuyang论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaRen, Yufei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYang, Han论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYu, Bin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China
- [12] Discovery of a potent and highly selective, orally efficacious IKK2 inhibitor for the treatment of rheumatoid arthritisABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Liddle, John论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Inc, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandWilliamson, Rick A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Inc, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Inc, Med Res Ctr, Stevenage SG1 2NY, Herts, England
- [13] Potent SMARCA2 targeted degraders induce genetic synthetic lethality in SMARCA4 deleted cancer.CANCER RESEARCH, 2021, 81 (13)Ito, Koichi论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAAgarwal, Anjana论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAPitis, Philip论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAWang, Min论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USACarter, Jack论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USACowart, Miles论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USADai, Chaofeng论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAGowen-MacDonald, William论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAElliot, Eliza论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAVidal, Brian论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USASpruance, Jacob论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USA论文数: 引用数: h-index:机构:Ruggeri, Bruce论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USALu, Liang论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USACombs, Andrew论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USALin, Hong论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAScherle, Peggy论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USAVaddi, Kris论文数: 0 引用数: 0 h-index: 0机构: Prelude Therapeut Inc, Wilmington, DE USA Prelude Therapeut Inc, Wilmington, DE USA
- [14] Selective PROTAC-mediated degradation of SMARCA2 is efficacious in SMARCA4 mutant cancersNature Communications, 13Jennifer Cantley论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Xiaofen Ye论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Emma Rousseau论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Tom Januario论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Brian D. Hamman论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Christopher M. Rose论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Tommy K. Cheung论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Trent Hinkle论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Leofal Soto论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Connor Quinn论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Alicia Harbin论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Elizabeth Bortolon论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Xin Chen论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Roy Haskell论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Eva Lin论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Shang-Fan Yu论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Geoff Del Rosario论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Emily Chan论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Debra Dunlap论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Hartmut Koeppen论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Scott Martin论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Mark Merchant论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Matt Grimmer论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Fabio Broccatelli论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Jing Wang论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Jennifer Pizzano论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Peter S. Dragovich论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Michael Berlin论文数: 0 引用数: 0 h-index: 0机构: Arvinas,Robert L. Yauch论文数: 0 引用数: 0 h-index: 0机构: Arvinas,
- [15] Discovery of a potent, highly selective, and orally efficacious small-molecule activator of the insulin receptorJOURNAL OF MEDICINAL CHEMISTRY, 2000, 43 (19) : 3487 - 3494Liu, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAXu, LB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USASzalkowski, D论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USALi, ZH论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USADing, V论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAKwei, G论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAHuskey, S论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAMoller, DE论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAHeck, JV论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAZhang, BB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAJones, AB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USA
- [16] Bifunctional Compounds as SMARCA2 Degraders for Treating CancerACS MEDICINAL CHEMISTRY LETTERS, 2021,Sabnis, Ram W.论文数: 0 引用数: 0 h-index: 0机构: Smith Gambrell & Russell LLP, Atlanta, GA 30309 USA Smith Gambrell & Russell LLP, Atlanta, GA 30309 USA
- [17] Selective PROTAC-mediated degradation of SMARCA2 is efficacious in SMARCA4 mutant cancersNATURE COMMUNICATIONS, 2022, 13 (01)Cantley, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAYe, Xiaofen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USARousseau, Emma论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAJanuario, Tom论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAHamman, Brian D.论文数: 0 引用数: 0 h-index: 0机构: HotSpot Therapeut & Nc, 1 Deerpk Dr,Ste C, Monmouth Jct, NJ 08852 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USARose, Christopher M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USACheung, Tommy K.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAHinkle, Trent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USASoto, Leofal论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAQuinn, Connor论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAHarbin, Alicia论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USABortolon, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAHaskell, Roy论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USALin, Eva论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAYu, Shang-Fan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USADel Rosario, Geoff论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAChan, Emily论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USADunlap, Debra论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAKoeppen, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAMartin, Scott论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAMerchant, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAGrimmer, Matt论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USABroccatelli, Fabio论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAWang, Jing论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAPizzano, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USADragovich, Peter S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USABerlin, Michael论文数: 0 引用数: 0 h-index: 0机构: Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USAYauch, Robert L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Arvinas LLC, 5 Sci Pk, New Haven, CT 06511 USA
- [18] Potent and orally efficacious PROTAC degraders of estrogen receptor α (ER α )CANCER RESEARCH, 2024, 84 (06)Rej, Rohan K.论文数: 0 引用数: 0 h-index: 0Chen, Zhixiang论文数: 0 引用数: 0 h-index: 0Acharyya, Ranjan K.论文数: 0 引用数: 0 h-index: 0Wu, Dimin论文数: 0 引用数: 0 h-index: 0Hu, Biao论文数: 0 引用数: 0 h-index: 0Xu, Guozhang论文数: 0 引用数: 0 h-index: 0Nagilla, Rakesh论文数: 0 引用数: 0 h-index: 0Metwally, Hoda论文数: 0 引用数: 0 h-index: 0Wang, Yu论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Bai, Longchuan论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [19] Discovery of Amino Alcohols as Highly Potent, Selective, and Orally Efficacious Inhibitors of Leukotriene A4 HydrolaseJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (23) : 16410 - 16425Thoma, Gebhard论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandMarkert, Christian论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandLueoend, Rainer论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandMiltz, Wolfgang论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandSpanka, Carsten论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandBollbuck, Birgit论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandWolf, Romain M.论文数: 0 引用数: 0 h-index: 0机构: Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandSrinivas, Honnappa论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharm AG, Chem Biol & Therapeut, Biomed Res, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandPenno, Carlos A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharm AG, Chem Biol & Therapeut, Biomed Res, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandKiffe, Michael论文数: 0 引用数: 0 h-index: 0机构: PK Sci Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandGajewska, Monika论文数: 0 引用数: 0 h-index: 0机构: PK Sci Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandBednarczyk, Dallas论文数: 0 引用数: 0 h-index: 0机构: Discovery & Translat Lab, Biomed Res, Novartis Pharm AG, Cambridge, MA 02139 USA Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandWieczorek, Grazyna论文数: 0 引用数: 0 h-index: 0机构: Immunol Dis Area, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandEvans, Amanda论文数: 0 引用数: 0 h-index: 0机构: Immunol Dis Area, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandBeerli, Christian论文数: 0 引用数: 0 h-index: 0机构: Immunol Dis Area, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, SwitzerlandRohn, Till A.论文数: 0 引用数: 0 h-index: 0机构: Immunol Dis Area, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland Global Discovery Chem, Biomed Res, Novartis Pharm AG, CH-4002 Basel, Switzerland
- [20] Discovery of Highly Potent, Selective, and Orally Efficacious p300/CBP Histone Acetyltransferases InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (03) : 1337 - 1360Yang, Yaxi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaZhang, Rukang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLi, Zhaojun论文数: 0 引用数: 0 h-index: 0机构: Dezhou Univ, Sch Informat Management, Dezhou 253023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaMei, Lianghe论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Suzhou Inst Drug Innovat, Shanghai Inst Mat Med, Suzhou 213000, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaWan, Shili论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaDing, Hong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaChen, Zhifeng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaXing, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaFeng, Huijin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaHan, Jie论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaJiang, Hualiang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaZheng, Mingyue论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaLuo, Cheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaZhou, Bing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Hangzhou Inst Adv Study, Beijing 100049, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, State Key Lab Drug Res, Shanghai 201203, Peoples R China