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- [1] Discovery of ERD-12310A as an Exceptionally Potent and Orally Efficacious PROTAC Degrader of Estrogen Receptor α (ERα)JOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (23) : 20933 - 20965Rej, Rohan Kalyan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAHu, Biao论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAChen, Zhixiang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAAcharyya, Ranjan Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWu, Dimin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMetwally, Hoda论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMceachern, Donna论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAJiang, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USABai, Longchuan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USANishimura, Leticia S.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAGersch, Christina L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Meilin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USACarlson, Kathryn论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Urbana, IL 61801 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAKatzenellenbogen, John A.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Urbana, IL 61801 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAXu, Guozhang论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 09406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAZhang, Weihong论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 09406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWu, Wenxue论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 09406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAPriestley, E. Scott论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 09406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 09406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USARae, James M.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Coll Pharm, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA
- [2] Discovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER plus Human Breast CancerJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (21) : 19010 - 19037Acharyya, Ranjan Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USARej, Rohan Kalyan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAHu, Biao论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAChen, Zhixiang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWu, Dimin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USALu, Jianfeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMetwally, Hoda论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMceachern, Donna论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAJiang, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USABai, Longchuan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USATosovic, Jelena论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAGersch, Christina L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAXu, Guozhang论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAZhang, Weihong论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWu, Wenxue论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAPriestley, E. Scott论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASarkari, Farzad论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USARae, James M.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Dept Pharmacol, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Internal Med, Dept Pharmacol,Div Hematol Oncol,Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA
- [3] Discovery of ERD-3111 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader with Strong Antitumor ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (17) : 12559 - 12585Chen, Zhixiang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAHu, Biao论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USARej, Rohan Kalyan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWu, Dimin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAAcharyya, Ranjan Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Mingliang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAXu, Tianfeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USALu, Jianfeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMetwally, Hoda论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAMceachern, Donna论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USABai, Longchuan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAGersch, Christina L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Meilin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAZhang, Wenjing论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USALi, Qiuxia论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USARae, James M.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Coll Pharm, Dept Med Chem, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA
- [4] Discovery of potent, highly selective and orally efficacious SMARCA2 degradersCANCER RESEARCH, 2024, 84 (06)Leng, Lingying论文数: 0 引用数: 0 h-index: 0Yang, Lin论文数: 0 引用数: 0 h-index: 0Tu, Wenbin论文数: 0 引用数: 0 h-index: 0Rej, Rohan论文数: 0 引用数: 0 h-index: 0Allu, Srinivasa Rao论文数: 0 引用数: 0 h-index: 0Huang, Liyue论文数: 0 引用数: 0 h-index: 0Jiang, Wei论文数: 0 引用数: 0 h-index: 0Wang, Yu论文数: 0 引用数: 0 h-index: 0Stuckey, Jeanne论文数: 0 引用数: 0 h-index: 0Sarkari, Farzad R.论文数: 0 引用数: 0 h-index: 0Wang, Meilin论文数: 0 引用数: 0 h-index: 0Wang, Lu论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [5] Discovery of Exceptionally Potent, Selective, and Efficacious PROTAC Degraders of CBP and p300 ProteinsJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (12) : 8178 - 8199Thomas, Junius Eugene论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAWang, Mi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAJiang, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAWang, Meilin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAWang, Lu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Program Chem Biol, Ann Arbor, MI 48104 USA
- [6] Identification and development of oral estrogen receptor PROTAC degraders for breast cancerCANCER RESEARCH, 2018, 78 (04)Flanagan, John J.论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USAQian, Yimin论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USAGough, Sheryl M.论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USAAndreoli, Monica论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USABookbinder, Mark论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USABradley, John论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USARousseau, Emma论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USAWillard, Ryan论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USACrews, Craig M.论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USACrew, Andrew P.论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USATaylor, Ian论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USAHouston, John论文数: 0 引用数: 0 h-index: 0机构: Arvinas Inc, New Haven, CT USA
- [7] The Quest for Orally Available Selective Estrogen Receptor Degraders (SERDs)CHEMMEDCHEM, 2020, 15 (22) : 2072 - 2097Wang, Lucia论文数: 0 引用数: 0 h-index: 0机构: Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07030 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07030 USA论文数: 引用数: h-index:机构:
- [8] Dynamics-Based Discovery of Novel, Potent Benzoic Acid Derivatives as Orally Bioavailable Selective Estrogen Receptor Degraders for ERα plus Breast CancerJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (11) : 7575 - 7595Zhang, Xiaomeng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Sanhome Pharmaceut Co Ltd, R&D Ctr, Nanjing 211135, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaWang, Yazhou论文数: 0 引用数: 0 h-index: 0机构: Nanjing Sanhome Pharmaceut Co Ltd, R&D Ctr, Nanjing 211135, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaLi, Xue论文数: 0 引用数: 0 h-index: 0机构: Nanjing Sanhome Pharmaceut Co Ltd, R&D Ctr, Nanjing 211135, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaWu, Jie论文数: 0 引用数: 0 h-index: 0机构: Nanjing Sanhome Pharmaceut Co Ltd, R&D Ctr, Nanjing 211135, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaZhao, Liwen论文数: 0 引用数: 0 h-index: 0机构: Nanjing Sanhome Pharmaceut Co Ltd, R&D Ctr, Nanjing 211135, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaLi, Wei论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaLiu, Jian论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China
- [9] New Class of Selective Estrogen Receptor Degraders (SERDs): Expanding the Toolbox of PROTAC DegronsACS MEDICINAL CHEMISTRY LETTERS, 2018, 9 (08): : 803 - 808Wang, Lucia论文数: 0 引用数: 0 h-index: 0机构: Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAGuillen, Valeria S.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USASharma, Naina论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAFlessa, Kevin论文数: 0 引用数: 0 h-index: 0机构: Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAMin, Jian论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USACarlson, Kathryn E.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAToy, Weiyi论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USABraqi, Sara论文数: 0 引用数: 0 h-index: 0机构: Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAKatzenellenbogen, Benita S.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAKatzenellenbogen, John A.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Chem, Dept Mol & Integrat Physiol, Urbana, IL 61801 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USAChandarlapaty, Sarat论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA Stevens Inst Technol, Dept Chem & Chem Biol, Hoboken, NJ 07601 USA论文数: 引用数: h-index:机构:
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