共 50 条
- [1] Discovery of Potent, Highly Selective, and Efficacious SMARCA2 DegradersJOURNAL OF MEDICINAL CHEMISTRY, 2024, 68 (02) : 1134 - 1154Li, Zhenwu论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAHarikrishnan, Lalgudi S.论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAXu, Guozhang论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USASamanta, Debangshu论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAClemente, Jose C.论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USALeng, Lingying论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USATu, Wenbin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAYang, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAWang, Mi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Med Sch, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Med Sch, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Coll Pharm, Dept Med Chem, Ann Arbor, MI 48109 USA SK Life Sci Labs, King Of Prussia, PA 19406 USADeng, Qiaolin论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USABehshad, Elham论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USANagilla, Rakesh论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAOrth, Peter论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USARice, Cory论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAStrickland, Corey论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAMohammad, Helai P.论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USAPriestley, E. Scott论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA SK Life Sci Labs, King Of Prussia, PA 19406 USA
- [2] Development of potent, highly selective and efficacious SMARCA2 degradersCANCER RESEARCH, 2024, 84 (06)Yang, Lin论文数: 0 引用数: 0 h-index: 0Tu, Wenbin论文数: 0 引用数: 0 h-index: 0Huang, Liyue论文数: 0 引用数: 0 h-index: 0Leng, Lingying论文数: 0 引用数: 0 h-index: 0Jiang, Wei论文数: 0 引用数: 0 h-index: 0Wang, Meilin论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Stuckey, Jeanne论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [3] Discovery of High-Affinity SMARCA2/4 Bromodomain Ligands and Development of Potent and Exceptionally Selective SMARCA2 PROTAC DegradersJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (02) : 1113 - 1133Leng, Lingying论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USATu, Wenbin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAYang, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Zhejiang Univ, Sir Run Shaw Hosp, Sch Med, Dept Pharmacol, Hangzhou 310058, Peoples R China Zhejiang Univ, Sir Run Shaw Hosp, Sch Med, Dept Pathol, Hangzhou 310058, Peoples R China Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Mi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAMeagher, Jennifer L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAChinnaswamy, Krishnapriya论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAAllu, Srinivasa Rao论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USARej, Rohan Kalyan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USATosovic, Jelena论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAHarikrishnan, Lalgudi论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USALi, Zhenwu论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAStuckey, Jeanne A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Dept Med Chem, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
- [4] Discovery of orally bioavailable SMARCA2/4 dual degraders for treatment of acute myeloid leukemiaCANCER RESEARCH, 2022, 82 (12)Abbineni, Chandrasekhar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKhare, Leena论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKuila, Bilash论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKhaji, Abdul Rawoof论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMahadeo, Dhaytadak Bhagwan论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDukare, Sandeep Vitthal论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKumar, Bhagya M. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGore, Suraj T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAhuja, Vijay Kamal论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDhudashiya, Amit A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRaghavendra, N. R.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGowda, Nagesh论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaCharamanna, K. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAithal, Kiran B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamiulla, D. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMukherjee, Subhendu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAntony, Thomas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGiri, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaChelur, Shekar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaNellore, Kavitha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDaginakatte, Girish论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRamachandra, Murali论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamajdar, Susanta论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India
- [5] Orally bioavailable SMARCA2 degraders with exceptional selectivity and potency.CANCER RESEARCH, 2021, 81 (13)Abbineni, Chandrasekhar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSatyam, Leena Khare论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKuila, Bilash论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaEttam, Ashok论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRawoof, Khaji Abdul论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSreevidya, M. R.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDukare, Sandeep Vitthal论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGore, Suraj T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaNankar, Rakesh P.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAhuja, Vijay Kamal论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaCharamanna, K. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGoyal, Megha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAithal, Kiran论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamiulla, D. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMukherjee, Subhendu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAntony, Thomas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGiri, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaChelur, Shekar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaNellore, Kavitha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDaginakatte, Girish论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRamachandra, Murali论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamajdar, Susanta论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India
- [6] Discovery of SMD-3236: A Potent, Highly Selective and Efficacious SMARCA2 Degrader for the Treatment of SMARC4-Deficient Human CancersJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (02) : 1155 - 1178Yang, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USATu, Wenbin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Coll Pharm, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USALeng, Lingying论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAJiang, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Mi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAMeagher, Jennifer L.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAChinnaswamy, Krishnapriya论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAStuckey, Jeanne A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Life Sci Inst, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Meilin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWen, Bo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USASun, Duxin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAHarikrishnan, Lalgudi论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAStrickland, Corey论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USARice, Cory论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAOrth, Peter论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: SK Life Sci Labs, King Of Prussia, PA 19406 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Coll Pharm, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA
- [7] Discovery of oral SMARCA2 degraders for the treatment of SMARCA4 mutant tumorsCANCER RESEARCH, 2024, 84 (06)Clemente, Jose C.论文数: 0 引用数: 0 h-index: 0Harikrishnan, Lal论文数: 0 引用数: 0 h-index: 0Knight, Steve论文数: 0 引用数: 0 h-index: 0Samanta, Debangshu论文数: 0 引用数: 0 h-index: 0Li, Zhenwu论文数: 0 引用数: 0 h-index: 0Nagilla, Rakesh论文数: 0 引用数: 0 h-index: 0Kendsersky, Nathan论文数: 0 引用数: 0 h-index: 0Joshi, Shreyas论文数: 0 引用数: 0 h-index: 0Orth, Peter论文数: 0 引用数: 0 h-index: 0Tudor, Matt论文数: 0 引用数: 0 h-index: 0Deng, Qiaolin论文数: 0 引用数: 0 h-index: 0Aguilar-Bonavides, Clemente论文数: 0 引用数: 0 h-index: 0Behshad, Elham论文数: 0 引用数: 0 h-index: 0Sui, Zhihua论文数: 0 引用数: 0 h-index: 0Strickland, Corey论文数: 0 引用数: 0 h-index: 0Jolivette, Larry J.论文数: 0 引用数: 0 h-index: 0Mohammad, Helai P.论文数: 0 引用数: 0 h-index: 0
- [8] Selective and orally bioavailable SMARCA2 targeted degraders induce synthetic lethality in SMARCA4-deficient solid tumorCANCER RESEARCH, 2023, 83 (07)Ito, Koichi论文数: 0 引用数: 0 h-index: 0Shvartsbart, Artem论文数: 0 引用数: 0 h-index: 0Rager, Joseph论文数: 0 引用数: 0 h-index: 0Agarwal, Anjana论文数: 0 引用数: 0 h-index: 0Hulse, Michael论文数: 0 引用数: 0 h-index: 0Vykuntam, Komali论文数: 0 引用数: 0 h-index: 0Wang, Min论文数: 0 引用数: 0 h-index: 0Kurian, Justin论文数: 0 引用数: 0 h-index: 0Cowart, Miles论文数: 0 引用数: 0 h-index: 0Cote, Joy论文数: 0 引用数: 0 h-index: 0Sivakumar, Monisha论文数: 0 引用数: 0 h-index: 0Carter, Jack论文数: 0 引用数: 0 h-index: 0Burtell, Jessica论文数: 0 引用数: 0 h-index: 0Grego, Alex论文数: 0 引用数: 0 h-index: 0Moore, Andrew论文数: 0 引用数: 0 h-index: 0Bhagwat, Neha论文数: 0 引用数: 0 h-index: 0Ruepp, Stefan论文数: 0 引用数: 0 h-index: 0Emme, Tom论文数: 0 引用数: 0 h-index: 0Lu, Liang论文数: 0 引用数: 0 h-index: 0Pitis, Philip论文数: 0 引用数: 0 h-index: 0Basch, Corey论文数: 0 引用数: 0 h-index: 0Bersch, Klare论文数: 0 引用数: 0 h-index: 0Mei, Song论文数: 0 引用数: 0 h-index: 0Leal, Raul论文数: 0 引用数: 0 h-index: 0Rose, John论文数: 0 引用数: 0 h-index: 0Roth, Danielle论文数: 0 引用数: 0 h-index: 0Cao, Ganfeng论文数: 0 引用数: 0 h-index: 0Vaddi, Kris论文数: 0 引用数: 0 h-index: 0Geeganage, Sandy论文数: 0 引用数: 0 h-index: 0Ruggeri, Bruce论文数: 0 引用数: 0 h-index: 0Combs, Andrew论文数: 0 引用数: 0 h-index: 0Scherle, Peggy论文数: 0 引用数: 0 h-index: 0
- [9] Preclinical characterization of PRT7732: A highly potent, selective, and orally bioavailable targeted protein degrader of SMARCA2CANCER RESEARCH, 2024, 84 (06)Shvartsbart, Artem论文数: 0 引用数: 0 h-index: 0Ito, Koichi论文数: 0 引用数: 0 h-index: 0Rager, Joseph论文数: 0 引用数: 0 h-index: 0Hulse, Michael论文数: 0 引用数: 0 h-index: 0Agarwal, Anjana论文数: 0 引用数: 0 h-index: 0Vykuntam, Komali论文数: 0 引用数: 0 h-index: 0Burtell, Jessica论文数: 0 引用数: 0 h-index: 0Wang, Min论文数: 0 引用数: 0 h-index: 0Kurian, Justin论文数: 0 引用数: 0 h-index: 0Cowart, Miles论文数: 0 引用数: 0 h-index: 0Cote, Joy论文数: 0 引用数: 0 h-index: 0Stahl, Nick论文数: 0 引用数: 0 h-index: 0Sivakumar, Monisha论文数: 0 引用数: 0 h-index: 0Reichelderfer, Anthony论文数: 0 引用数: 0 h-index: 0Carter, Jack论文数: 0 引用数: 0 h-index: 0Grego, Alexander论文数: 0 引用数: 0 h-index: 0Moore, Andrew论文数: 0 引用数: 0 h-index: 0Bhagwat, Neha论文数: 0 引用数: 0 h-index: 0Kuskovsky, Ross论文数: 0 引用数: 0 h-index: 0Ganesan, Shanthi论文数: 0 引用数: 0 h-index: 0Ruepp, Stefan论文数: 0 引用数: 0 h-index: 0Emm, Tom论文数: 0 引用数: 0 h-index: 0Pitis, Philip论文数: 0 引用数: 0 h-index: 0Basch, Corey论文数: 0 引用数: 0 h-index: 0Bersch, Klare论文数: 0 引用数: 0 h-index: 0Pan, Yongchun论文数: 0 引用数: 0 h-index: 0Mei, Song论文数: 0 引用数: 0 h-index: 0Leal, Raul论文数: 0 引用数: 0 h-index: 0Rose, John论文数: 0 引用数: 0 h-index: 0Roth, Dani论文数: 0 引用数: 0 h-index: 0Xu, Chaoyi论文数: 0 引用数: 0 h-index: 0Cao, Ganfeng论文数: 0 引用数: 0 h-index: 0Vaddi, Kris论文数: 0 引用数: 0 h-index: 0Lee, Sang Hyun论文数: 0 引用数: 0 h-index: 0Geeganage, Sandy论文数: 0 引用数: 0 h-index: 0Combs, Andrew论文数: 0 引用数: 0 h-index: 0Scherle, Peggy论文数: 0 引用数: 0 h-index: 0
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