SYNTHESIS AND STRUCTURE ELUCIDATION OF BENZOTHIAZOLE-CONTAINING COMPOUNDS FOR ANTIMICROBIAL INVESTIGATION

被引：0

作者：

GHONEIM, KM ^{[1
]}

ELBASIL, S ^{[1
]}

OSMAN, AN ^{[1
]}

SAID, MM ^{[1
]}

MEGAHED, SA ^{[1
]}

机构：

[1] UNIV CAIRO,FAC PHARM,DEPT MICROBIOL,CAIRO,EGYPT

来源：

REVUE ROUMAINE DE CHIMIE | 1991年 / 36卷 / 11-12期

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Attempted cycloaddition of benzimidazole-2-thiol with arylidenemalononitriles 1 was unsuccessful. 2-Cyanomethyl-1,3-benzothiazole 6 condensed with certain aromatic aldehydes to produce 7, cycloaddition of which with cyanoacethydrazide 3 yielded B. Structure of the newly synthesized compounds was substantiated by spectroscopic data and/or unambiguous synthesis. Representative compounds were screened for antimicrobial activity.

引用

页码：1355 / 1361

页数：7

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