Solvent-free microwave assisted synthesis of (E)-1-{3-[2-(9-Ethyl-9H-carbazol-3-yl)vinyl]benzofuran-2-yl}-2,2-dimethylpropan-1-ones and their antimicrobial activity

被引：8

作者：

Ashok, D. ^{[1
]}

Sidda, Ravi ^{[1
]}

Lakshmi, B. Vijaya ^{[1
]}

Ganesh, Arram ^{[1
]}

机构：

[1] Osmania Univ, Dept Chem, Hyderabad 500007, Andhra Pradesh, India

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2014年 / 84卷 / 11期

关键词：

microwave assisted synthesis; carbazole-3-carbaldehyde; carbazolylaryl prop-2-enones; carbazolylvinylbenzofurans; antimicrobial activity; CHALCONES; DERIVATIVES; BENZOFURAN;

D O I：

10.1134/S1070363214110280

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

We report the solvent-free synthesis of (E)-1-{3-[2-(9-Ethyl-9H-carbazol-3-yl)vinyl]benzofuran-2-yl}-2,2-dimethylpropan-1-ones starting with 9-Ethyl-9H-carbazole-3-carbaldehyde under conventional and microwave irradiation methods. All products were characterised by IR, H-1 NMR, C-13 NMR, mass spectrometry, and elemental analysis. The compounds were tested in vitro for their antimicrobial activity.

引用

页码：2211 / 2217

页数：7

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