Solvent-free microwave assisted synthesis of (E)-1-{3-[2-(9-Ethyl-9H-carbazol-3-yl)vinyl]benzofuran-2-yl}-2,2-dimethylpropan-1-ones and their antimicrobial activity

被引：8
|
作者：
Ashok, D. [1 ]
Sidda, Ravi [1 ]
Lakshmi, B. Vijaya [1 ]
Ganesh, Arram [1 ]
机构：
[1] Osmania Univ, Dept Chem, Hyderabad 500007, Andhra Pradesh, India
来源：
RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2014年 / 84卷 / 11期
关键词：
microwave assisted synthesis; carbazole-3-carbaldehyde; carbazolylaryl prop-2-enones; carbazolylvinylbenzofurans; antimicrobial activity; CHALCONES; DERIVATIVES; BENZOFURAN;
D O I：
10.1134/S1070363214110280
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
We report the solvent-free synthesis of (E)-1-{3-[2-(9-Ethyl-9H-carbazol-3-yl)vinyl]benzofuran-2-yl}-2,2-dimethylpropan-1-ones starting with 9-Ethyl-9H-carbazole-3-carbaldehyde under conventional and microwave irradiation methods. All products were characterised by IR, H-1 NMR, C-13 NMR, mass spectrometry, and elemental analysis. The compounds were tested in vitro for their antimicrobial activity.
引用
收藏
页码：2211 / 2217
页数：7
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