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- [32] Discovery of highly potent and selective orexin 1 receptor antagonists (1-SORAs) suitable for in vivo interrogation of orexin 1 receptor pharmacologyBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (23) : 5809 - 5814Stump, Craig A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USACooke, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USABruno, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Vitro Pharmacol, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USACabalu, Tamara D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Pharmacokinet Pharmacodynam & Drug Metab, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAGotter, Anthony L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAHarell, C. Meacham论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAKuduk, Scott D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAMcDonald, Terrence P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAO'Brien, Julie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Vitro Pharmacol, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USARenger, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAWilliams, Peter D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAWinrow, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurosci, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USAColeman, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, West Point, PA 19486 USA Merck Res Labs, Discovery Chem, West Point, PA 19486 USA
- [33] Discovery of 3,9-diazabicyclo[4.2.1]nonanes as potent dual orexin receptor antagonists with sleep-promoting activity in the ratBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (14) : 4201 - 4205Coleman, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USASchreier, John D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARoecker, Anthony J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMercer, Swati P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcGaughey, Georgia B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Modeling & Informat, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USACox, Christopher D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHartman, George D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHarrell, C. Meacham论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAReiss, Duane R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USADoran, Scott M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGarson, Susan L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAAnderson, Wayne B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USATang, Cuyue论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAPrueksaritanont, Thomayant论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAWinrow, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARenger, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Depress & Circadian Disorders, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA
- [34] PHARMACOLOGICAL CHARACTERIZATION OF OREXIN RECEPTOR ANTAGONISTSSLEEP, 2011, 34 : A5 - A5Winrow, C. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USADoran, S. M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAGotter, A. L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAPausch, M. H.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAKuduk, S. D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAUslaner, J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USACarroll, S. S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USASmith, S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USAColeman, P. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USARenger, J. J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA USA Merck Res Labs, West Point, PA USA
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