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- [21] Effectiveness of analogs of the kappa opioid receptor antagonist (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic) to reduce U50,488-induced diuresis and stress-induced cocaine reinstatement in ratsPSYCHOPHARMACOLOGY, 2010, 210 (02) : 189 - 198Beardsley, Patrick M.论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth Univ, Sch Med, Dept Pharmacol & Toxicol, Richmond, VA 23284 USA VCU Inst Drug & Alcohol Studies, Richmond, VA USA Virginia Commonwealth Univ, Sch Med, Dept Pharmacol & Toxicol, Richmond, VA 23284 USAPollard, Gerald T.论文数: 0 引用数: 0 h-index: 0机构: Howard Associates LLC, Res Triangle Pk, NC USA Virginia Commonwealth Univ, Sch Med, Dept Pharmacol & Toxicol, Richmond, VA 23284 USAHoward, James L.论文数: 0 引用数: 0 h-index: 0机构: Howard Associates LLC, Res Triangle Pk, NC USA Virginia Commonwealth Univ, Sch Med, Dept Pharmacol & Toxicol, Richmond, VA 23284 USACarroll, F. Ivy论文数: 0 引用数: 0 h-index: 0机构: Res Triangle Inst, Res Triangle Pk, NC 27709 USA Virginia Commonwealth Univ, Sch Med, Dept Pharmacol & Toxicol, Richmond, VA 23284 USA
- [22] Effectiveness of analogs of the kappa opioid receptor antagonist (3R)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic) to reduce U50,488-induced diuresis and stress-induced cocaine reinstatement in ratsPsychopharmacology, 2010, 210 : 189 - 198Patrick M. Beardsley论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth University,Department of Pharmacology and Toxicology, School of MedicineGerald T. Pollard论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth University,Department of Pharmacology and Toxicology, School of MedicineJames L. Howard论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth University,Department of Pharmacology and Toxicology, School of MedicineF. Ivy Carroll论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth University,Department of Pharmacology and Toxicology, School of Medicine
- [23] Crystal structure of 1-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydrofuran-2-yl)-2-propylsulfanyl-1H-pyrimidin-4-one, C12H18N2O5SZEITSCHRIFT FUR KRISTALLOGRAPHIE-NEW CRYSTAL STRUCTURES, 2009, 224 (01): : 107 - 108Euler, Harald论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, Germany Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, GermanyKirfel, Armin论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, Germany Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, GermanyEl-Tayeb, Ali论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, PharmaCtr Bonn, Inst Pharmaceut, D-53121 Bonn, Germany Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, GermanyMueller, Christa E.论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, PharmaCtr Bonn, Inst Pharmaceut, D-53121 Bonn, Germany Univ Bonn, Mineral Petrol Inst, D-53115 Bonn, Germany
- [24] Discovery of (2S)-8[(3R)-3-Methylmorpholin-4-yl]-1-(3-methyl-2-oxobutyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido[1,2-a]pyrimidin-6-one: A Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid TumorsJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (01) : 376 - 400Pasquier, Benoit论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceEl-Ahmad, Youssef论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceFiloche-Romme, Bruno论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceDureuil, Christine论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceFassy, Florence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceAbecassis, Pierre-Yves论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Drug Disposit & Safety, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMathieu, Magali论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBertrand, Thomas论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBenard, Tsiala论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Pharmaceut Sci Operat, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBarriere, Cedric论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceEl Batti, Samira论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLetallec, Jean-Philippe论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceSonnefraud, Veronique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBrollo, Maurice论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceDelbarre, Laurence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLoyau, Veronique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FrancePilorge, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBertin, Luc论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceRichepin, Patrick论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceArigon, Jerome论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLabrosse, Jean-Robert论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceClement, Jacques论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceDurand, Florence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceCombet, Romain论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FrancePerraut, Pierre论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLeroy, Vincent论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceGay, Frederic论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLefrancois, Dominique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBretin, Francois论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMarquette, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMichot, Nadine论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Prot Prod, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceCaron, Anne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Global Biotherapeut, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceCastell, Christelle论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceSchio, Laurent论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMcCort, Gary论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceGoulaouic, Helene论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceGarcia-Echeverria, Carlos论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceRonan, Baptiste论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France
- [25] Identification of (R)-6-(1-(4-Cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro-1H-pyrazol-3-yl)-2-methoxynicotinic Acid, a Highly Potent and Selective Nonsteroidal Mineralocorticoid Receptor AntagonistJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (10) : 4273 - 4288Casimiro-Garcia, Agustin论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAPiotrowski, David W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAAmbler, Catherine论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAArhancet, Graciela B.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Med Chem, Chesterfield, MO 63017 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USABanker, Mary Ellen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USABanks, Tereece论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USABoustany-Kari, Carine M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USACai, Cuiman论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAChen, Xiangyang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Med Chem, Chesterfield, MO 63017 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAEudy, Rena论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAHepworth, David论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAHulford, Catherine A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAJennings, Sandra M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USALoria, Paula M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAMeyers, Marvin J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Med Chem, Chesterfield, MO 63017 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAPetersen, Donna N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USARaheja, Neil K.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USASammons, Matthew论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Cambridge, MA 02139 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAShe, Li论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USASong, Kun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Cambridge, MA 02139 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAVrieze, Derek论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USAWei, Liuqing论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Cambridge, MA 02140 USA
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USAGoldenblatt, Peter论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Vitro Pharmacol, 33 Ave Louis Pasteur, Boston, MA 02115 USA Merck & Co Inc, Dept Med Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USAShaffer, Lynse论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Vitro Pharmacol, 33 Ave Louis Pasteur, Boston, MA 02115 USA Merck & Co Inc, Dept Med Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USAPatel, San Ita B.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Struct Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USA Merck & Co Inc, Dept Med Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USALesburg, Charles A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Struct Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USA Merck & Co Inc, Dept Med Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USAAlpert, Carla论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Vitro Pharmacol, 33 Ave Louis Pasteur, Boston, MA 02115 USA Merck & Co Inc, Dept Med Chem, 33 Ave Louis Pasteur, Boston, MA 02115 USADorosh, 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