A VERSATILE APPROACH TO 2,3-DISUBSTITUTED INDOLES THROUGH THE PALLADIUM-CATALYZED CYCLIZATION OF ORTHO-ALKYNYLTRIFLUOROACETANILIDES WITH VINYL TRIFLATES AND ARYL HALIDES

被引：0

作者：

ARCADI, A

CACCHI, S

MARINELLI, F

机构：

[1] UNIV LAQUILA,DIPARTIMENTO CHIM INGN CHIM & MAT,V ASSERGI 4,I-67100 LAQUILA,ITALY

[2] UNIV ROME LA SAPIENZA,DIPARTIMENTO STUDI CHIM & TECNOL SOSTANZE BIOLOGICAMENTE ATT V,I-00185 ROME,ITALY

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 27期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The Palladium-catalyzed cyclization of o-alkynyltrifluoroacetanilides with vinyl triflates and aryl halides produces 2,3-disubstituted indoles in good to high yield.

引用

页码：3915 / 3918

页数：4

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