A VERSATILE APPROACH TO 2,3-DISUBSTITUTED INDOLES THROUGH THE PALLADIUM-CATALYZED CYCLIZATION OF ORTHO-ALKYNYLTRIFLUOROACETANILIDES WITH VINYL TRIFLATES AND ARYL HALIDES

被引：0
|
作者：
ARCADI, A
CACCHI, S
MARINELLI, F
机构：
[1] UNIV LAQUILA,DIPARTIMENTO CHIM INGN CHIM & MAT,V ASSERGI 4,I-67100 LAQUILA,ITALY
[2] UNIV ROME LA SAPIENZA,DIPARTIMENTO STUDI CHIM & TECNOL SOSTANZE BIOLOGICAMENTE ATT V,I-00185 ROME,ITALY
来源：
TETRAHEDRON LETTERS | 1992年 / 33卷 / 27期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The Palladium-catalyzed cyclization of o-alkynyltrifluoroacetanilides with vinyl triflates and aryl halides produces 2,3-disubstituted indoles in good to high yield.
引用
收藏
页码：3915 / 3918
页数：4
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