BIOCHEMICAL-CHARACTERIZATION OF SR48692, A SELECTIVE NONPEPTIDE ANTAGONIST OF THE NEUROTENSIN RECEPTOR

被引:0
|
作者
OURYDONAT, F [1 ]
HEAULME, M [1 ]
THURNEYSSEN, O [1 ]
GONALONS, N [1 ]
GULLY, D [1 ]
LEFUR, G [1 ]
SOUBRIE, P [1 ]
机构
[1] SANOFI RECH,F-34082 MONTPELLIER,FRANCE
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:U122 / U122
页数:1
相关论文
共 50 条
  • [21] EFFECTS OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST SR 48692 ON RAT AND GUINEA-PIG GI MOTILITY
    CROCI, T
    LANDI, M
    MANARA, L
    GULLY, D
    LEFUR, G
    GASTROENTEROLOGY, 1995, 108 (04) : A958 - A958
  • [22] SR-48692 - Antipsychotic - Neurotensin antagonist
    不详
    DRUGS OF THE FUTURE, 2001, 26 (12) : 1217 - 1217
  • [23] Neurotensin Receptor 1 Antagonist SR48692 Improves Response to Carboplatin by Enhancing Apoptosis and Inhibiting Drug Efflux in Ovarian Cancer
    Liu, Jin
    Agopiantz, Mikael
    Poupon, Joel
    Wu, Zherui
    Just, Pierre-Alexandre
    Borghese, Bruno
    Segal-Bendirdjian, Evelyne
    Gauchotte, Guillaume
    Gompel, Anne
    Forgez, Patricia
    CLINICAL CANCER RESEARCH, 2017, 23 (21) : 6516 - 6528
  • [24] [H-3]SR-48692, THE FIRST NONPEPTIDE NEUROTENSIN ANTAGONIST RADIOLIGAND CHARACTERIZATION OF BINDING-PROPERTIES AND EVIDENCE FOR DISTINCT AGONIST AND ANTAGONIST BINDING DOMAINS ON THE RAT NEUROTENSIN RECEPTOR
    LABBEJULLIE, C
    BOTTO, JM
    MAS, MV
    CHABRY, J
    MAZELLA, J
    VINCENT, JP
    GULLY, D
    MAFFRAND, JP
    KITABGI, P
    MOLECULAR PHARMACOLOGY, 1995, 47 (05) : 1050 - 1056
  • [25] Neurotensin receptor-1 antagonist SR48692 modulation of high-fat diet-induced pathogenesis of NAFLD in mice
    Pal, Himanshu
    Verma, Pradeep
    Mohanty, Banalata
    EUROPEAN JOURNAL OF LIPID SCIENCE AND TECHNOLOGY, 2024, 126 (06)
  • [26] Neurotensin receptor-1 antagonist SR48692 modulation of high-fat diet induced reproductive impairment in male mice
    Verma, Pradeep
    Pal, Himanshu
    Mohanty, Banalata
    REPRODUCTIVE TOXICOLOGY, 2024, 123
  • [27] The neurotensin receptor antagonist SR 48692, decreases extracellular striatal GABA in rats
    Chapman, MA
    See, RE
    BRAIN RESEARCH, 1996, 729 (01) : 124 - 126
  • [28] A Machine-Assisted Flow Synthesis of SR48692: A Probe for the Investigation of Neurotensin Receptor-1
    Battilocchio, Claudio
    Deadman, Benjamin J.
    Nikbin, Nikzad
    Kitching, Matthew O.
    Baxendale, Ian R.
    Ley, Steven V.
    CHEMISTRY-A EUROPEAN JOURNAL, 2013, 19 (24) : 7917 - 7930
  • [29] The Specific Neurotensin Receptor (ntr1) Antagonist, Sr48692, Sensitizes Prostate Cancer Cells to Ionizing Radiation, in Both In Vitro and In Vivo Models
    Larner, J. M.
    Dziegielewski, J.
    Pemberton, B.
    Dunlap-Brown, M.
    Parsons, S.
    Amorino, G.
    INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 2009, 75 (03): : S561 - S561
  • [30] Neurotensin receptor-mediated inhibition of pancreatic cancer cell growth by the neurotensin antagonist SR 48692
    Herzig, MCS
    Chapman, WG
    Sheridan, A
    Rake, JB
    Woynarowski, JM
    ANTICANCER RESEARCH, 1999, 19 (1A) : 213 - 219