EFFECTS OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST SR 48692 ON RAT AND GUINEA-PIG GI MOTILITY

被引:0
|
作者
CROCI, T
LANDI, M
MANARA, L
GULLY, D
LEFUR, G
机构
[1] SANOFI MIDY SPA,RES CTR,I-20137 MILAN,ITALY
[2] SANOFI RECH,F-31036 TOULOUSE,FRANCE
[3] SANOFI RECH,F-75008 PARIS,FRANCE
关键词
D O I
10.1016/0016-5085(95)28136-3
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
引用
收藏
页码:A958 / A958
页数:1
相关论文
共 50 条
  • [1] SR-48692, A NONPEPTIDE NEUROTENSIN RECEPTOR ANTAGONIST, BLOCKS THE CARDIOVASCULAR EFFECTS ELICITED BY NEUROTENSIN IN GUINEA-PIGS
    NISATO, D
    GUIRAUDOU, P
    BARTHELEMY, G
    GULLY, D
    LEFUR, G
    LIFE SCIENCES, 1994, 54 (07) : PL95 - PL100
  • [2] DIFFERENTIAL-EFFECTS OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST, SR-48692, ON THE PHARMACOLOGICAL EFFECTS OF NEUROTENSIN AGONISTS
    PUGSLEY, TA
    AKUNNE, HC
    WHETZEL, SZ
    DEMATTOS, S
    CORBIN, AE
    WILEY, JN
    WUSTROW, DJ
    WISE, LD
    HEFFNER, TG
    PEPTIDES, 1995, 16 (01) : 37 - 44
  • [3] EFFECT OF THE NONPEPTIDE NEUROTENSIN ANTAGONIST, SR-48692, AND 2 ENANTIOMERIC ANALOGS, SR-48527 AND SR-49711, ON NEUROTENSIN BINDING AND CONTRACTILE RESPONSES IN GUINEA-PIG ILEUM AND COLON
    LABBEJULLIE, C
    DESCHAINTRES, S
    GULLY, D
    LEFUR, G
    KITABGI, P
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1994, 271 (01): : 267 - 276
  • [4] EFFECTS OF NEUROTENSIN ON GUINEA-PIG INTESTINAL MOTILITY
    YAU, WM
    NEMETH, PR
    GASTROENTEROLOGY, 1977, 72 (05) : 1153 - 1153
  • [5] THE NONPEPTIDE NEUROTENSIN ANTAGONIST, SR-48692 USED AS A TOOL TO REVEAL PUTATIVE NEUROTENSIN RECEPTOR SUBTYPES
    DUBUC, I
    COSTENTIN, J
    TERRANOVA, JP
    BARNOUIN, MC
    SOUBRIE, P
    LEFUR, G
    ROSTENE, W
    KITABGI, P
    BRITISH JOURNAL OF PHARMACOLOGY, 1994, 112 (02) : 352 - 354
  • [6] BIOCHEMICAL-CHARACTERIZATION OF SR48692, A SELECTIVE NONPEPTIDE ANTAGONIST OF THE NEUROTENSIN RECEPTOR
    OURYDONAT, F
    HEAULME, M
    THURNEYSSEN, O
    GONALONS, N
    GULLY, D
    LEFUR, G
    SOUBRIE, P
    BRITISH JOURNAL OF PHARMACOLOGY, 1994, 112 : U122 - U122
  • [7] Inhibition of neurotensin-induced pancreatic carcinoma growth by a nonpeptide neurotensin receptor antagonist, SR48692
    Iwase, K
    Evers, BM
    Hellmich, MR
    Kim, HJ
    Higashide, S
    Gully, D
    Thompson, JC
    Townsend, CM
    CANCER, 1997, 79 (09) : 1787 - 1793
  • [8] INCREASE IN NEUROTENSIN RECEPTOR EXPRESSION IN RAT-BRAIN INDUCED BY CHRONIC TREATMENT WITH THE NONPEPTIDE NEUROTENSIN RECEPTOR ANTAGONIST SR-48692
    AZZI, M
    NICOT, A
    GULLY, D
    KITABGI, P
    BEROD, A
    ROSTENE, W
    NEUROSCIENCE LETTERS, 1994, 172 (1-2) : 97 - 100
  • [9] THE NONPEPTIDE NK-2 ANTAGONIST SR 48968 IS ALSO A NK-3 ANTAGONIST IN THE GUINEA-PIG BUT NOT IN THE RAT
    PETITET, F
    BEAUJOUAN, JC
    SAFFROY, M
    TORRENS, Y
    GLOWINSKI, J
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1993, 191 (01) : 180 - 187
  • [10] SR-48692 - Antipsychotic - Neurotensin antagonist
    不详
    DRUGS OF THE FUTURE, 2001, 26 (12) : 1217 - 1217