APPEARANCE OF PHYSICAL-DEPENDENCE AND ANALGESIC ACTIVITY OF 2-(5H-[1]-BENZOPYRANO[2,3-B]PYRIDIN-7-YL)PROPIONIC ACID (Y-8004) BY REPEATED ADMINISTRATION

被引：2
|
作者：
MARUYAMA, Y [1 ]
ANAMI, K [1 ]
IMAYOSHI, T [1 ]
IMAMURA, H [1 ]
机构：
[1] YOSHITOMI PHARMACEUT IND LTD, RES LABS, FUKUOKA 871, JAPAN
来源：
YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN | 1977年 / 97卷 / 04期
关键词：
D O I：
10.1248/yakushi1947.97.4_343
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：343 / 349
页数：7
相关论文
共 44 条
  • [31] Synthesis, single crystal x-ray analysis, and antimicrobial activity of new (22E)-N'-(4-methoxybenzylidene)-2-[3-cyano-7,8-dihydro-4-(5-methylfuran-2-yl)-2-oxo-2H-pyrano[4,3-b]pyridin-1(5H)-yl]acetohydrazide
    Amr, A. E.
    Mohamed, S. F.
    Al-Omar, M. A.
    Ghabbour, H. A.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2016, 86 (07) : 1758 - 1761
  • [32] Synthesis, single crystal x-ray analysis, and antimicrobial activity of new (22E)-N'-(4-methoxybenzylidene)-2-[3-cyano-7,8-dihydro-4-(5-methylfuran-2-yl)-2-oxo-2H-pyrano[4,3-b]pyridin-1(5H)-yl]acetohydrazide
    A. E. Amr
    S. F. Mohamed
    M. A. Al-Omar
    H. A. Ghabbour
    Russian Journal of General Chemistry, 2016, 86 : 1758 - 1761
  • [33] Improving the Pharmacokinetic and CYP Inhibition Profiles of Azaxanthene-Based Glucocorticoid Receptor Modulators-Identification of (S)-5-(2-(9-Fluoro-2-(4-(2-hydroxypropan-2-yl)phenyl)-5H-chromeno[2,3-b]pyridin-5-yl)-2-methylpropanamido)-N-(tetrahydro-2H-pyran-4-yl)-1,3,4-thiadiazole-2-carboxamide (BMS-341)
    Yang, Michael G.
    Dhar, T. G. Murali
    Xiao, Zili
    Xiao, Hai-Yun
    Duan, James J. -W.
    Jiang, Bin
    Galella, Michael A.
    Cunningham, Mark
    Wang, Jinhong
    Habte, Sium
    Shuster, David
    McIntyre, Kim W.
    Carman, Julie
    Holloway, Deborah A.
    Somerville, John E.
    Nadler, Steven G.
    Salter-Cid, Luisa
    Barrish, Joel C.
    Weinstein, David S.
    JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (10) : 4278 - 4290
  • [34] PHARMACOKINETIC BEHAVIOR IN POLYMORPHONUCLEAR LEUKOCYTES OF N,N-DIMETHYLCARBAMOYLMETHYL ALPHA,2-DIMETHYL-5H-[1]BENZOPYRANO[2,3-B]-PYRIDINE-7-ACETATE (Y-23023), A NEW PRODRUG TYPE OF ANTIINFLAMMATORY AGENT, AND INDOMETHACIN AFTER ORAL ADMINISTRATIONS IN RATS
    YAMADA, I
    NAGAMATSU, Y
    IMAYOSHI, T
    SHIBATA, M
    TSUJI, A
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 1994, 46 (07) : 614 - 616
  • [35] Discovery of 1-[3-(1-Methyl-1H-pyrazol-4-y1)-5-oxo-5H-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl]-N-(pyridin-2-ylmethyl)methanesulfonamide (MK-8033): A Specific c-Met/Ron Dual Kinase Inhibitor with Preferential Affinity for the Activated State of c-Met
    Northrup, Alan B.
    Katcher, Matthew H.
    Altman, Michael D.
    Chenard, Melissa
    Daniels, Matthew H.
    Deshmukh, Sujal V.
    Falcone, Danielle
    Guerin, David J.
    Hatch, Harold
    Li, Chaomin
    Lu, Wei
    Lutterbach, Bart
    Allison, Timothy J.
    Patel, Sangita B.
    Reily, John F.
    Reutershan, Michael
    Rickert, Keith W.
    Rosenstein, Craig
    Soisson, Stephen M.
    Szewczak, Alexander A.
    Walker, Deborah
    Wilson, Kevin
    Young, Jonathan R.
    Pan, Bo-Sheng
    Dinsmore, Christopher J.
    JOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (06) : 2294 - 2310
  • [36] COMPOUNDS WITH POTENTIAL ACTIVITY AGAINST GASTRIC-SECRETION AND GASTRIC-ULCERS .4. SYNTHESIS OF 3-PHENYL-2-OXO-5-[2-(4-METHYLPIPERAZIN-1-YL)-ACETYL]-1H-2,3,4,5-TETRAHYDROPYRIDO[2,3-B][1,4]DIAZEPINE
    BIANCHI, M
    BUTTI, A
    FARMACO-EDIZIONE SCIENTIFICA, 1984, 39 (02): : 162 - 170
  • [37] Novel alpha-amino-3-hydroxy-5-methylisoxazole-4-propionate receptor antagonists: Synthesis and structure-activity relationships of 6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-pyrido[2,3-b]pyrazinedione and related compounds
    Ohmori, J
    Kubota, H
    ShimizuSasamata, M
    Okada, M
    Sakamoto, S
    JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (06) : 1331 - 1338
  • [38] Potent platelet-derived growth factor-β receptor (PDGF-βR) inhibitors:: Synthesis and structure-activity relationships of 7-[3-(cyclohexylmethyl)ureido]-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl}quinoxalin-2(1H)-one derivatives
    Aoki, Katsuyuki
    Obata, Tatsuhiro
    Yamazaki, Yosuke
    Mori, Yoshikazu
    Hirokawa, Hiroko
    Koseki, Jun-ichi
    Hattori, Tomohisa
    Niitsu, Kazuaki
    Takeda, Shuichi
    Aburanda, Masaki
    Miyamoto, Ken-ichi
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2007, 55 (02) : 255 - 267
  • [39] Domino reactions in the synthesis of benzothieno[2,3-c]pyridines. New one-pot method of preparing 2-([1]benzothieno-[2,3-c]pyridin-1-yl)benzoic acids and 8,13b-dihydro[1]benzothieno[2′,3′:3,4]pyrido-[2,1-a]isoindol-5(7H)-ones
    Tolkunov, V. S.
    Eres'ko, A. B.
    Khizhan, A. I.
    Mazepa, A. V.
    Palamarchuk, G. V.
    Shishkin, O. V.
    Tolkunov, S. V.
    CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2012, 48 (04) : 666 - 671
  • [40] Domino reactions in the synthesis of benzothieno[2,3-c]pyridines. New one-pot method of preparing 2-([1]benzothieno-[2,3-c]pyridin-1-yl)benzoic acids and 8,13b-dihydro[1]benzothieno[2',3':3,4]pyrido-[2,1-a]isoindol-5(7 H)-ones
    V. S. Tolkunov
    A. B. Eres’ko
    A. I. Khizhan
    A. V. Mazepa
    G. V. Palamarchuk
    O. V. Shishkin
    S. V. Tolkunov
    Chemistry of Heterocyclic Compounds, 2012, 48 : 666 - 671
12345