X-ray Structure for an RNase H Inhibitor Bound to HIV-1 Reverse Transcriptase
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作者:
Himmel, Daniel M.
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Rutgers State Univ, CABM, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Himmel, Daniel M.
[1
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Sarafianos, Stefan G.
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Rutgers State Univ, CABM, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Sarafianos, Stefan G.
[1
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Dharmasena, Sanjeewa
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机构:
Univ Pittsburgh, Sch Med, Pittsburgh, PA 15260 USARutgers State Univ, CABM, New Brunswick, NJ USA
Dharmasena, Sanjeewa
[2
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Hossain, Mofazzal
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Univ Pittsburgh, Sch Med, Pittsburgh, PA 15260 USARutgers State Univ, CABM, New Brunswick, NJ USA
Hossain, Mofazzal
[2
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McCoy-Simandle, Kessler
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Univ Pittsburgh, Sch Med, Pittsburgh, PA 15260 USARutgers State Univ, CABM, New Brunswick, NJ USA
McCoy-Simandle, Kessler
[2
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Clark, Patrick K.
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NCI, Frederick Canc Res & Dev Ctr, Bethesda, MD 20892 USARutgers State Univ, CABM, New Brunswick, NJ USA
Clark, Patrick K.
[3
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Clark, Arthur D., Jr.
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Rutgers State Univ, CABM, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Clark, Arthur D., Jr.
[1
]
Knight, Jennifer L.
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Rutgers State Univ, Dept Chem & Chem Biol, New Brunswick, NJ USA
Rutgers State Univ, BIOMAPS Inst Quantitat Biol, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Knight, Jennifer L.
[4
,5
]
Levy, Ronald M.
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机构:
Rutgers State Univ, Dept Chem & Chem Biol, New Brunswick, NJ USA
Rutgers State Univ, BIOMAPS Inst Quantitat Biol, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Levy, Ronald M.
[4
,5
]
Hughes, Stephen H.
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NCI, Frederick Canc Res & Dev Ctr, Bethesda, MD 20892 USARutgers State Univ, CABM, New Brunswick, NJ USA
Hughes, Stephen H.
[3
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Parniak, Michael A.
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Univ Pittsburgh, Sch Med, Pittsburgh, PA 15260 USARutgers State Univ, CABM, New Brunswick, NJ USA
Parniak, Michael A.
[2
]
Arnold, Eddy
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Rutgers State Univ, CABM, New Brunswick, NJ USARutgers State Univ, CABM, New Brunswick, NJ USA
Arnold, Eddy
[1
]
机构:
[1] Rutgers State Univ, CABM, New Brunswick, NJ USA
[2] Univ Pittsburgh, Sch Med, Pittsburgh, PA 15260 USA
[3] NCI, Frederick Canc Res & Dev Ctr, Bethesda, MD 20892 USA
[4] Rutgers State Univ, Dept Chem & Chem Biol, New Brunswick, NJ USA
[5] Rutgers State Univ, BIOMAPS Inst Quantitat Biol, New Brunswick, NJ USA
来源:
ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES
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2005年
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61卷
关键词:
HIV-1 reverse transcriptase;
RNase H inhibitor;
rational inhibitor design;
机构:Univ Rochester, Infect Dis Unit, Dept Med, Sch Med & Dent, Rochester, NY 14642 USA
Wang, Jiong
Bambara, Robert A.
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Univ Rochester, Dept Biochem & Biophys, Sch Med & Dent, Rochester, NY 14642 USAUniv Rochester, Infect Dis Unit, Dept Med, Sch Med & Dent, Rochester, NY 14642 USA
Bambara, Robert A.
Demeter, Lisa M.
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机构:Univ Rochester, Infect Dis Unit, Dept Med, Sch Med & Dent, Rochester, NY 14642 USA
Demeter, Lisa M.
Dykes, Carrie
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Univ Rochester, Infect Dis Unit, Dept Med, Sch Med & Dent, Rochester, NY 14642 USAUniv Rochester, Infect Dis Unit, Dept Med, Sch Med & Dent, Rochester, NY 14642 USA
机构:
Seoul Natl Univ, Coll Pharm, Seoul, South Korea
Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul, South KoreaSeoul Natl Univ, Coll Pharm, Seoul, South Korea
Lee, J. S.
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Hattori, M.
Kim, J.
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Seoul Natl Univ, Coll Pharm, Seoul, South Korea
Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul, South KoreaSeoul Natl Univ, Coll Pharm, Seoul, South Korea
机构:
Seoul Natl Univ, Coll Pharm, Seoul 151742, South Korea
Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 151742, South KoreaSeoul Natl Univ, Coll Pharm, Seoul 151742, South Korea
Lee, Ji Suk
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Hattori, Masao
Kim, Jinwoong
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Seoul Natl Univ, Pharmaceut Sci Res Inst, Seoul 151742, South KoreaSeoul Natl Univ, Coll Pharm, Seoul 151742, South Korea
机构:
Ultrafast Optical Processes Laboratory, Department of Chemistry, University of PennsylvaniaUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Kuroda D.G.
Bauman J.D.
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Center for Advanced Biotechnology and Medicine, Piscataway
Department of Chemistry and Chemical Biology, Rutgers University, PiscatawayUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Bauman J.D.
Challa J.R.
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Ultrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Department of Chemistry, University of Rochester, RochesterUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Challa J.R.
Patel D.
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Center for Advanced Biotechnology and Medicine, Piscataway
Department of Medicinal Chemistry, Rutgers University, PiscatawayUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Patel D.
Troxler T.
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Ultrafast Optical Processes Laboratory, Department of Chemistry, University of PennsylvaniaUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Troxler T.
Das K.
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Center for Advanced Biotechnology and Medicine, Piscataway
Department of Chemistry and Chemical Biology, Rutgers University, PiscatawayUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Das K.
Arnold E.
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Center for Advanced Biotechnology and Medicine, Piscataway
Department of Chemistry and Chemical Biology, Rutgers University, Piscataway
Department of Medicinal Chemistry, Rutgers University, PiscatawayUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
Arnold E.
Hochstrasser R.M.
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Ultrafast Optical Processes Laboratory, Department of Chemistry, University of PennsylvaniaUltrafast Optical Processes Laboratory, Department of Chemistry, University of Pennsylvania
机构:
CUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USACUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
Zhang, Baofeng
D'Erasmo, Michael P.
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CUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
CUNY, Grad Ctr, PhD Program Chem, New York, NY 10016 USACUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
D'Erasmo, Michael P.
Murelli, Ryan P.
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CUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
CUNY, Grad Ctr, PhD Program Chem, New York, NY 10016 USACUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
Murelli, Ryan P.
Gallicchio, Emilio
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CUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA
CUNY, Grad Ctr, PhD Program Chem, New York, NY 10016 USA
CUNY, Grad Ctr, PhD Program Biochem, New York, NY 10016 USACUNY, Brooklyn Coll, Dept Chem, 2900 Bedford Ave, Brooklyn, NY 11210 USA