共 50 条
- [31] MEDI 20-Discovery and characterization of allosteric inhibitors of Bcr-Abl kinaseABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 236Gray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA
- [32] MEDI 190-Discovery of Fms/Kit kinase inhibitors for the treatment of rheumatoid arthritisABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232Bremer, Ryan论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZhang, Jiazhong论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAWu, Guoxian论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZhou, Yong论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAOh, Angela论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Biol Struct, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAShellooe, Rafe论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Prot Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USACheung, Ivana论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Assay Dev & Screening, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAEng, Kevin论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Mol Biol, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USABurton, Betsy论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Assay Dev & Screening, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USALuu, Catherine论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Prot Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USANespi, Marika论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZhu, Hongyao论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Informat, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USATabrizizad, Maryam论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Biol Struct, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USADe Joya-Rice, Julie论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Assay Dev & Screening, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZhang, Kam论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Biol Struct, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAHurt, Clarence论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USASpevak, Wayne论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZuckerman, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Biol Struct, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAZhang, Chao论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Informat, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAPowell, Ben论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Prot Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAHabets, Gaston论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Assay Dev & Screening, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAWest, Brian论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Assay Dev & Screening, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USABollag, Gideon论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Div Discovery Biol, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAArtis, D. Rick论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Div Lead Generat, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USAIbrahim, Prabha论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA Plexxikon Inc, Dept Chem, Berkeley, CA 94706 USA
- [33] MEDI 233-Discovery and chiral synthesis of potent c-Met (HGFR) aminopyridine inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234Kung, Pei-Pei论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Med Chem, PGRD, San Diego, CA 92121 USA Pfizer, Dept Med Chem, PGRD, San Diego, CA 92121 USA
- [34] Discovery and optimization of orally active cyclohexane-based prolylcarboxypeptidase (PrCP) inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (23) : 6228 - 6233Debenham, John S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGraham, Thomas H.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAVerras, Andreas论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZhang, Yong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAClements, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKuethe, Jeffrey T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Proc Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMadsen-Duggan, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALiu, Wensheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USABhatt, Urmi R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, Dunlu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, Qing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGarcia-Calvo, Margarita论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGeissler, Wayne M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHe, Huaibing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALi, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALisnock, JeanMarie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept In Vitro Sci, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShen, Zhu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATong, Xinchun论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATung, Elaine C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAWiltsie, Judyann论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept In Vitro Sci, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAXu, Suoyu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHale, Jeffrey J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAPinto, Shirly论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShen, Dong-Ming论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [35] Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (01) : 140 - 152论文数: 引用数: h-index:机构:Cleghorn, Laura A. T.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandMcElroy, Stuart P.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandRobinson, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandSmith, Victoria C.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland论文数: 引用数: h-index:机构:Harrison, Justin R.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandNorcross, Neil R.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandSpinks, Daniel论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandBayliss, Tracy论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandNorval, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandStojanovski, Laste论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandTorrie, Leah S.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandFrearson, Julie A.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandBrenk, Ruth论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandFairlamb, Alan H.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandFerguson, Michael A. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandRead, Kevin D.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandWyatt, Paul G.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, ScotlandGilbert, Ian H.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Drug Discovery Unit, Div Biol Chem & Drug Discovery, Coll Life Sci,Sir James Black Ctr, Dundee DD1 5EH, Scotland
- [36] Discovery of triazines as potent, selective and orally active PDE4 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (15) : 4308 - 4314Gewald, Rainer论文数: 0 引用数: 0 h-index: 0机构: BioCrea GmbH, D-01445 Radebeul, Germany BioCrea GmbH, D-01445 Radebeul, GermanyGrunwald, Christian论文数: 0 引用数: 0 h-index: 0机构: BioCrea GmbH, D-01445 Radebeul, Germany BioCrea GmbH, D-01445 Radebeul, GermanyEgerland, Ute论文数: 0 引用数: 0 h-index: 0机构: BioCrea GmbH, D-01445 Radebeul, Germany BioCrea GmbH, D-01445 Radebeul, Germany
- [37] Recent advances in the discovery of small molecule c-Met Kinase inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 143 : 1103 - 1138Parikh, Palak K.论文数: 0 引用数: 0 h-index: 0机构: Nirma Univ, Inst Pharm, Dept Pharmaceut Chem, Ahmadabad 382481, Gujarat, India Nirma Univ, Inst Pharm, Dept Pharmaceut Chem, Ahmadabad 382481, Gujarat, IndiaGhate, Manjunath D.论文数: 0 引用数: 0 h-index: 0机构: Nirma Univ, Inst Pharm, Dept Pharmaceut Chem, Ahmadabad 382481, Gujarat, India Nirma Univ, Inst Pharm, Dept Pharmaceut Chem, Ahmadabad 382481, Gujarat, India
- [38] Discovery, optimization and biological evaluation for novel c-Met kinase inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 143 : 491 - 502Yuan, Haoliang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Inst Pharmaceut Res, Jiangsu Key Lab Drug Discovery Metab Dis, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaLiu, Qiufeng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, Key Lab Receptor Res, Shanghai 201203, Peoples R China ShanghaiTech Univ, Sch Life Sci & Technol, Shanghai 200031, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaZhang, Li论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaHu, Shihe论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaChen, Tiantian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, Key Lab Receptor Res, Shanghai 201203, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaLi, Huifang论文数: 0 引用数: 0 h-index: 0机构: Univ British Columbia, Vancouver Prostate Ctr, 2660 Oak St, Vancouver, BC V6H 3Z6, Canada China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaChen, Yadong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaXu, Yechun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, Key Lab Receptor Res, Shanghai 201203, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R ChinaLu, Tao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Inst Pharmaceut Res, Jiangsu Key Lab Drug Discovery Metab Dis, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China
- [39] Discovery of 6-benzyloxyquinolines as c-Met selective kinase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (04) : 1405 - 1409Nishii, Hiroki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanChiba, Takashi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanMorikami, Kenji论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Discovery Platform Technol, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanFukami, Takaaki A.论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Discovery Platform Technol, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanSakamoto, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Pharmaceut Res 2, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanKo, Kwangseok论文数: 0 引用数: 0 h-index: 0机构: C&C Res Labs, Hwaseong Si 445380, Gyeonggi Do, South Korea Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, JapanKoyano, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Dept Chem Res 2, Kamakura, Kanagawa 2478530, Japan
- [40] Discovery and optimization of triazolopyridazines as potent and selective inhibitors of the c-Met kinaseJOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (10) : 2879 - 2882Albrecht, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAHarmange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABauer, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABerry, Loren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABode, Christiane论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USABoezio, Alessandro A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAChen, April论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAChoquette, Deborah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USADussault, Isabelle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USAFridrich, Cary论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAHirai, Satoko论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAHoffman, Doug论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USALarrow, Jay F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAKaplan-Lefko, Paula论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USALin, Jasmine论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USALohman, Julia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USALong, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAMoriguchi, Jodi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USAO'Connor, Anne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAPotashman, Michele H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAReese, Monica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USARex, Karen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USASiegmund, Aaron论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USAShah, Kavita论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAShimanovich, Roman论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USASpringer, Stephanie K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USATeffera, Yohannes论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USAZhang, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Cambridge, MA 02139 USABellon, Steven F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA 02139 USA Amgen Inc, Cambridge, MA 02139 USA