Cyclocondensation of methyl 2-(1,3-benzothiazol-2-ylimino)-3,3,3-trifluoropropionate with C,N-binucleophiles

被引：0
|
作者：
Sokolov, V. B. [1 ]
Aksinenko, A. Yu. [1 ]
机构：
[1] Russian Acad Sci, Inst Physiologically Act Subst, Chernogolovka 142432, Moscow Oblast, Russia
来源：
RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2011年 / 81卷 / 05期
基金：
俄罗斯基础研究基金会;
关键词：
Trione; Exocyclic Nitrogen Atom; Trifluoropropionate; Ylimino;
D O I：
10.1134/S1070363211050161
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Reactions of methyl 2-(1,3-benzothiazol-2-ylimino)-3,3,3-trifluoropropionate with 1,3-C,N-binucleophiles, methyl 2-aminobut-2-enoate, 2-aminobut-2-enenitrile and N-substituted 6-aminouracils and 3-aminocyclohex-2-en-1-ones, led to the formation of trifluoromethyl-substituted heterocycles, dihydro-1H-pyrroles, hexahydro-1H-pyrrolo[2,3-d]pyrimidine-2,4,6-triones, and hexahydro-1H-indole-2,4-diones.
引用
收藏
页码：934 / 936
页数：3
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