Influence of the reaction conditions in the N-alkylation of acridone-2-carboxylic acids

被引：0
|
作者：
Marill, LX [1 ]
Comdom, RFP [1 ]
Hermández, MM [1 ]
机构：
[1] Ctr Pharmaceut Chem, Havana, Cuba
来源：
SYNTHETIC COMMUNICATIONS | 2001年 / 31卷 / 14期
关键词：
D O I：
10.1081/SCC-100104467
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis and a study about the influence of the solvent in the alkylation reaction of 2-Carboxy-6-chloro-9(10H) acridone (3b) and 2-Carboxy-6-chloro-7-nitro-9(10H) acridone (3a) was done, obtaining the N-ethyl ester derivative of the alkylated products. Using the liquid-liquid phase transfer catalysis only the N-alkylated derivative was obtained in both cases with an improved yield.
引用
收藏
页码：2159 / 2167
页数：9
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