Hypervalent iodine(III) sulfonate mediated synthesis of imidazo[1,2-a]pyridines

被引:10
|
作者
Huang, HY
Hou, RS
Wang, HM
Chen, LC [1 ]
机构
[1] Kaohsiung Med Univ, Grad Inst Pharmaceut Sci, Kaohsiung 807, Taiwan
[2] Chung Hwa Coll Med Technol, Tainan 717, Taiwan
关键词
hypervalent iodine(III) sulfonate; cyclocondensation; 2-aminopyridines;
D O I
10.1002/jccs.200400201
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
A direct and efficient method for the conversion of alkyl aryl ketones to imidazo[1,2-a]pyridines has been developed based on initial formation of alpha-organosulfonyloxy ketones and their subsequent cyclocondensation by 2-aminopyridines in one-pot conditions.
引用
收藏
页码:1377 / 1380
页数:4
相关论文
共 50 条
  • [41] Recent Advances in the Synthesis of Imidazo[1,2-a]pyridines: A Brief Review
    Panda, Jasmine
    Raiguru, Bishnu P. P.
    Mishra, Mitali
    Mohapatra, Seetaram
    Nayak, Sabita
    CHEMISTRYSELECT, 2022, 7 (03):
  • [42] FACILE SYNTHESIS OF IMIDAZO[1,2-a]PYRIDINES VIA TANDEM REACTION
    Jia, Jiong
    Ge, Yan-Qing
    Tao, Xu-Tang
    Wang, Jian-Wu
    HETEROCYCLES, 2010, 81 (01) : 185 - 194
  • [43] Synthesis of imidazo[1,2-a]pyridines from α,β-unsaturated aldehydes (microreview)
    Natalia A. Keiko
    Nadezhda V. Vchislo
    Chemistry of Heterocyclic Compounds, 2016, 52 : 222 - 224
  • [44] One-step synthesis of imidazo[1,2-a]pyridines in water
    Zali-Boeini, H.
    Norastehfar, N.
    Rudbari, H. Amiri
    RSC ADVANCES, 2016, 6 (85) : 81943 - 81949
  • [45] Metal-Free Synthesis of Trifluoromethyl Carbinol-Containing Imidazo[1,2-a ]pyridines via Dehydrative Coupling of Imidazo[1,2-a ]pyridines with Trifluoroacetaldehyde
    Liu, Zhaowen
    Guo, Xiaohua
    Chen, Zhixi
    Wu, Longhui
    Yang, Kai
    SYNTHESIS-STUTTGART, 2024, 56 (11): : 1756 - 1764
  • [46] Electrochemical oxidative iodination of imidazo[1,2-a]pyridines using NaI as iodine source
    Park, Jin Wha
    Kim, Yong Hwan
    Kim, Dae Young
    SYNTHETIC COMMUNICATIONS, 2020, 50 (05) : 710 - 718
  • [47] Copper-Mediated Aerobic Oxidative Synthesis of 3-Bromo-imidazo[1,2-a]pyridines with Pyridines and Enamides
    Zhou, Xiaoqiang
    Yan, Hao
    Ma, Chaowei
    He, Yongqin
    Li, Yamin
    Cao, Jinhui
    Yan, Rulong
    Huang, Guosheng
    JOURNAL OF ORGANIC CHEMISTRY, 2016, 81 (01): : 25 - 31
  • [48] Solvent-dependence of KI Mediated Electrosynthesis of Imidazo[1,2-a]pyridines
    Yi, Yangjie
    Xu, Leitao
    Liu, Yuyang
    Li, Mingfang
    Zhang, Lijuan
    Ye, Jiao
    Hu, Aixi
    CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2023, 39 (02) : 318 - 324
  • [49] Solvent-dependence of KI Mediated Electrosynthesis of Imidazo[1,2-a]pyridines
    Yangjie Yi
    Leitao Xu
    Yuyang Liu
    Mingfang Li
    Lijuan Zhang
    Jiao Ye
    Aixi Hu
    Chemical Research in Chinese Universities, 2023, 39 : 318 - 324