Hypervalent iodine(III) sulfonate mediated synthesis of imidazo[1,2-a]pyridines

被引：10
|
作者：
Huang, HY
Hou, RS
Wang, HM
Chen, LC [1 ]
机构：
[1] Kaohsiung Med Univ, Grad Inst Pharmaceut Sci, Kaohsiung 807, Taiwan
[2] Chung Hwa Coll Med Technol, Tainan 717, Taiwan
来源：
JOURNAL OF THE CHINESE CHEMICAL SOCIETY | 2004年 / 51卷 / 06期
关键词：
hypervalent iodine(III) sulfonate; cyclocondensation; 2-aminopyridines;
D O I：
10.1002/jccs.200400201
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A direct and efficient method for the conversion of alkyl aryl ketones to imidazo[1,2-a]pyridines has been developed based on initial formation of alpha-organosulfonyloxy ketones and their subsequent cyclocondensation by 2-aminopyridines in one-pot conditions.
引用
收藏
页码：1377 / 1380
页数：4
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