Structure-based discovery of non-peptidic small molecule inhibitors of Caspase-3

被引：0
|
作者：
Sakai, J
Yoshimori, A
Takasawa, R
Tanuma, SI
机构：
[1] Tokyo Univ Sci, Dept Biochem, Chiba, Japan
[2] Tokyo Univ Sci, Genome & Drug Res Ctr, Chiba, Japan
[3] Tokyo Univ Sci, Res Inst Biol Sci, Chiba, Japan
[4] Inst Theoret Med Inc, Tokyo, Japan
来源：
FEBS JOURNAL | 2005年 / 272卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：522 / 522
页数：1
相关论文
共 50 条
  • [31] Correction: Discovery of novel non-peptidic and non-covalent small-molecule 3CLpro inhibitors as potential candidate for COVID-19 treatment
    Zhidong Jiang
    Bo Feng
    Yumin Zhang
    Tianqing Nie
    Hong Liu
    Jia Li
    Haixia Su
    Leike Zhang
    Yi Zang
    Yu Zhou
    Signal Transduction and Targeted Therapy, 8
  • [32] Non-Peptidic Small Molecule Components from Cone Snail Venoms
    Lin, Zhenjian
    Torres, Joshua P.
    Watkins, Maren
    Paguigan, Noemi
    Niu, Changshan
    Imperial, Julita S.
    Tun, Jortan
    Safavi-Hemami, Helena
    Finol-Urdaneta, Rocio K.
    Neves, Jorge L. B.
    Espino, Samuel
    Karthikeyan, Manju
    Olivera, Baldomero M.
    Schmidt, Eric W.
    FRONTIERS IN PHARMACOLOGY, 2021, 12
  • [33] Structure-based virtual screening against SARS-3CLpro to identify novel non-peptidic hits
    Mukherjee, Prasenjit
    Desai, Prashant
    Ross, Larry
    White, E. Lucile
    Avery, Mitchell A.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (07) : 4138 - 4149
  • [34] Non-peptidic small-molecule inhibitors of the single-chain hepatitis C virus NS3 protease/NS4A cofactor complex discovered by structure-based NMR screening
    Wyss, DF
    Arasappan, A
    Senior, MM
    Wang, YS
    Beyer, BM
    Njoroge, FG
    McCoy, MA
    JOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (10) : 2486 - 2498
  • [35] Identification of potent and novel small-molecule inhibitors of caspase-3
    Allen, DA
    Pham, P
    Choong, IC
    Fahr, B
    Burdett, MT
    Lew, W
    DeLano, WL
    Gordon, EM
    Lam, JW
    O'Brien, T
    Lee, D
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (21) : 3651 - 3655
  • [36] Structure-based discovery of new selective small-molecule sirtuin 5 inhibitors
    Liu, Sha
    Ji, Sen
    Yu, Zhu-Jun
    Wang, Hua-Li
    Cheng, Xu
    Li, Wei-Jian
    Jing, Li
    Yu, Yamei
    Chen, Qiang
    Yang, Ling-Ling
    Li, Guo-Bo
    Wu, Yong
    CHEMICAL BIOLOGY & DRUG DESIGN, 2018, 91 (01) : 257 - 268
  • [37] Structure-Based Discovery of Small-Molecule Inhibitors of the Autocatalytic Proliferation of α-Synuclein Aggregates
    Chia, Sean
    Brotzakis, Z. Faidon
    Horne, Robert I.
    Possenti, Andrea
    Mannini, Benedetta
    Cataldi, Rodrigo
    Nowinska, Magdalena
    Staats, Roxine
    Linse, Sara
    Knowles, Tuomas P. J.
    Habchi, Johnny
    Vendruscolo, Michele
    MOLECULAR PHARMACEUTICS, 2022, : 183 - 193
  • [38] Recent progress in the drug discovery of non-peptidic BACE1 inhibitors
    Hamada, Yoshio
    Kiso, Yoshiaki
    EXPERT OPINION ON DRUG DISCOVERY, 2009, 4 (04) : 391 - 416
  • [39] 3,4-Dihydropyrimido(1,2-a)indol-10(2H)-ones as potent non-peptidic inhibitors of caspase-3
    Havran, Lisa M.
    Chong, Dan C.
    Childers, Wayne E.
    Dollings, Paul J.
    Dietrich, Arlene
    Harrison, Boyd L.
    Marathias, Vasilios
    Tawa, Gregory
    Aulabaugh, Ann
    Cowling, Rebecca
    Kapoor, Bhupesh
    Xu, Weixin
    Mosyak, Lidia
    Moy, Franklin
    Hum, Wah-Tung
    Wood, Andrew
    Robichaud, Albert J.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (22) : 7755 - 7768
  • [40] The initial evaluation of non-peptidic small-molecule HDM2 inhibitors based on p53-HDM2 complex structure
    Zhao, JH
    Wang, MJ
    Chen, J
    Luo, AP
    Wang, XQ
    Wu, M
    Yin, DL
    Liu, ZH
    CANCER LETTERS, 2002, 183 (01) : 69 - 77
12345