Pyrrolidine-fused iminoheterocycles as BACE1 inhibitors for the treatment of Alzheimer's disease

被引:0
|
作者
Gilbert, Eric [1 ]
Huang, Chunli [1 ]
Stamford, Andrew [1 ]
Cumming, Jared [1 ]
Greenlee, William [1 ]
Kennedy, Matthew [2 ]
Parker, Eric [2 ]
Kuvelkar, Reshma [3 ]
Cox, Kathleen [5 ]
Voight, Johannes [4 ]
Strickland, Corey [6 ]
Palamanda, Jairam [5 ]
机构
[1] Merck Res Labs, Dept Chem, Rahway, NJ 07065 USA
[2] Merck Res Labs, Dept CNS Biol, Kenilworth, NJ 07033 USA
[3] Merck Res Labs, Dept In Vitro Sci, Kenilworth, NJ 07033 USA
[4] Merck Res Labs, Dept Chem Modeling & Informat, Rahway, NJ 07065 USA
[5] Merck Res Labs, Dept Exploratory Drug Metab, Kenilworth, NJ 07033 USA
[6] Merck Res Labs, Dept Struct Chem, Kenilworth, NJ 07033 USA
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
101-MEDI
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页数:1
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