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- [41] A first-in-human, open-label, phase I trial of daily oral PCLX-001, an NMT inhibitor, in patients with relapsed/refractory B-cell lymphomas and advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2023, 41 (16)Sangha, Randeep S.论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaJamal, Rahima论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaSpratlin, Jennifer L.论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaKuruvilla, John论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaSehn, Laurie Helen论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaWeickert, Michael论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaBerthiaume, Luc G.论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, CanadaMackey, John Robert论文数: 0 引用数: 0 h-index: 0机构: Cross Canc Inst, Edmonton, AB, Canada
- [42] First-in-Human Phase I/IB Dose-Finding Study of Adagrasib (MRTX849) in Patients With Advanced KRASG12C Solid Tumors (KRYSTAL-1)JOURNAL OF CLINICAL ONCOLOGY, 2022, 40 (23) : 2530 - +Ou, Sai-Hong Ignatius论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Sch Med, Orange, CA 92868 USA Univ Calif Irvine, Chao Family Comprehens Canc Ctr, Orange, CA 92868 USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Lowe Ctr Thorac Oncol, Dana Farber Canc Inst, Boston, MA 02115 USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USALeal, Ticiana A.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, Madison, WI USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USARybkin, Igor I.论文数: 0 引用数: 0 h-index: 0机构: Henry Ford Canc Inst, Detroit, MI USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USASabari, Joshua K.论文数: 0 引用数: 0 h-index: 0机构: New York Univ Langone Hlth, Perlmutter Canc Ctr, New York, NY USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USABarve, Minal A.论文数: 0 引用数: 0 h-index: 0机构: Mary Crowley Canc Ctr, Dallas, TX USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USABazhenova, Lyudmila论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Moores Canc Ctr, La Jolla, CA 92093 USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAJohnson, Melissa L.论文数: 0 引用数: 0 h-index: 0机构: Tennessee Oncol, Sarah Cannon Res Inst, Nashville, TN USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAVelastegui, Karen L.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut Inc, San Diego, CA USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USACilliers, Cornelius论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut Inc, San Diego, CA USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAChristensen, James G.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut Inc, San Diego, CA USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAYan, Xiaohong论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut Inc, San Diego, CA USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAChao, Richard C.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut Inc, San Diego, CA USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: START San Antonio, San Antonio, TX USA Univ Calif Irvine, Sch Med, Orange, CA 92868 USA
- [43] Results of the first-in-human phase I trial assessing MSC2156119J (EMD 1214063), an oral selective c-Met inhibitor, in patients (pts) with advanced solid tumorsJOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Falchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAHong, David S.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAAmin, Hesham M.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAFu, Siqing论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAPiha-Paul, Sarina Anne论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAJanku, Filip论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAGranda, J. Gabrielle论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAZheng, Hongxia论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAKlevesath, Manfred B.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAKoehler, Karola论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USABladt, Friedhelm论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAJohne, Andreas论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USAKurzrock, Razelle论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Invest Canc Therapeut, Phase Clin Trials Program 1, Houston, TX 77030 USA
- [44] BPI-9016M, a novel c-Met inhibitor, in pretreated advanced solid tumor: Results from a first-in-human, phase I, dose-escalation study.JOURNAL OF CLINICAL ONCOLOGY, 2018, 36 (15)Hu, Xingsheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaZheng, Xin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaMo, Hongnan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaCui, Xinge论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaDing, Lieming论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaTan, Fenlai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaHu, Pei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R ChinaShi, Yuankai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Beijing Key Lab Clin Study Anticancer Mol Targete, Canc Hosp, Natl Canc Ctr, Beijing, Peoples R China
- [45] First-in-human biomarker-driven phase I TRESR trial of ataxia telangiectasia and Rad3related inhibitor (ATRi) RP-3500 in patients (pts) with advanced solid tumors harboring synthetic lethal (SL) genomic alterationsMOLECULAR CANCER THERAPEUTICS, 2021, 20 (12)Yap, Timothy论文数: 0 引用数: 0 h-index: 0Lee, Elizabeth论文数: 0 引用数: 0 h-index: 0Spigel, David论文数: 0 引用数: 0 h-index: 0Fontana, Elisa论文数: 0 引用数: 0 h-index: 0Hojgaard, Martin论文数: 0 引用数: 0 h-index: 0Lheureux, Stephanie论文数: 0 引用数: 0 h-index: 0Mettu, Niharika B.论文数: 0 引用数: 0 h-index: 0Carter, Louise论文数: 0 引用数: 0 h-index: 0Plummer, Ruth论文数: 0 引用数: 0 h-index: 0Ulanet, Danielle论文数: 0 引用数: 0 h-index: 0Manley, Peter论文数: 0 引用数: 0 h-index: 0Jiang, Ying论文数: 0 引用数: 0 h-index: 0Rosen, Ezra论文数: 0 引用数: 0 h-index: 0
- [46] Preliminary safety, antitumor activity, and circulating tumor DNA (ctDNA) changes with RMC-9805, an oral, RAS(ON) G12D-selective tri-complex inhibitor in patients with KRAS G12D pancreatic ductal adenocarcinoma (PDAC) from a phase 1 study in advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2025, 43 (4_SUPPL) : 724 - 724Spira, Alexander I.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAKim, Dae Won论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAParikh, Aparna Raj论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USABarve, Minal A.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAPowderly, John D.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAStarodub, Alexander论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAStrickler, John H.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USALi, Bob T.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAOberstein, Paul Eliezer论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAHassan, Faisal论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAYang, Michelle论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAMccleland, Mark论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USALally, Satwant论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USALin, Wei论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USASohoni, Sophia论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USAHong, David S.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists Res Inst, Fairfax, VA USA
- [47] Preliminary phase I results from a first-in-human study of EMB-02, a PD-1xLAG-3 bispecific antibody, in patients (pts) with advanced solid tumorsANNALS OF ONCOLOGY, 2023, 34 : S625 - S625Day, D.论文数: 0 引用数: 0 h-index: 0机构: Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, Australia Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaGanju, V.论文数: 0 引用数: 0 h-index: 0机构: Peninsula & Southeast Oncol, Oncol Dept, Frankston, Vic, Australia Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaChung, K.论文数: 0 引用数: 0 h-index: 0机构: Prisma Hlth Syst Upstate GHS Canc Inst, Oncol, Greenville, SC USA Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaSi, L.论文数: 0 引用数: 0 h-index: 0机构: Peking Univ Canc Hosp & Inst, Dept Renal Canc & Melanoma, Beijing, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaMao, L.论文数: 0 引用数: 0 h-index: 0机构: Peking Univ Canc Hosp & Inst, Dept Renal Canc & Melanoma, Beijing, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaAghmesheh, M.论文数: 0 引用数: 0 h-index: 0机构: Southern Med Day Care Ctr, Med Oncol Dept, Wollongong, NSW, Australia Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaHoyer, R.论文数: 0 引用数: 0 h-index: 0机构: Mem Hosp Cent, Med Oncol Dept, UCHlth Canc Care & Hematol Clin, Colorado Springs, CO USA Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaBrewin, K.论文数: 0 引用数: 0 h-index: 0机构: Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, Australia Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaZeng, S.论文数: 0 引用数: 0 h-index: 0机构: Shanghai EpimAb Biotherapeut Co Ltd, Clin Dev, Shanghai, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaLu, Q.论文数: 0 引用数: 0 h-index: 0机构: Shanghai EpimAb Biotherapeut Co Ltd, Clin Dev, Shanghai, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaJiang, C.论文数: 0 引用数: 0 h-index: 0机构: Shanghai EpimAb Biotherapeut Co Ltd, Clin Dev, Shanghai, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaRen, F.论文数: 0 引用数: 0 h-index: 0机构: Shanghai EpimAb Biotherapeut Co Ltd, Clin Dev, Shanghai, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaWu, X.论文数: 0 引用数: 0 h-index: 0机构: Shanghai EpimAb Biotherapeut Co Ltd, Biol Dept, Shanghai, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, AustraliaGuo, J.论文数: 0 引用数: 0 h-index: 0机构: Peking Univ Canc Hosp & Inst, Dept Renal Canc & Melanoma, Beijing, Peoples R China Monash Hlth, Med Oncol Dept, Monash Med Ctr, Clayton, Vic, Australia
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