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- [31] Trial in progress: A phase Ib study of AMG 510, a specific and irreversible KRASG12C inhibitor, in combination with other anticancer therapies in patients with advanced solid tumors harboring KRAS p.G12C mutation (CodeBreak 101).JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (15)Fakih, Marwan论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USADurm, Greg Andrew论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USAGovindan, Ramaswamy论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USAFalchook, Gerald Steven论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USASoman, Neelesh论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USAHenary, Haby Adel论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USAHong, David S.论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, 1500 E Duarte Rd, Duarte, CA 91010 USA
- [32] A phase 1 clinical trial to evaluate safety, tolerability, pharmacokinetics (PK) and efficacy of D-1553, a novel KRASG12C inhibitor, in patients with advanced or metastatic solid tumor harboring KRASG12C mutation.CANCER RESEARCH, 2022, 82 (12)Price, Timothy论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaGrewal, Jaspreet论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, AustraliaAbed, Afaf论文数: 0 引用数: 0 h-index: 0机构: Norton Canc Inst, Louisville, KY USA Linear Clin Res Ltd, Nedlands, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaMoore, Melissa论文数: 0 引用数: 0 h-index: 0机构: St Vincents Hosp Melbourne, Fitzroy, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaYeh, Yu-Min论文数: 0 引用数: 0 h-index: 0机构: Natl Cheng Kung Univ Hosp, Tainan, Taiwan Queen Elizabeth Hosp TQEH, Woodville South, AustraliaGadgeel, Shirish论文数: 0 引用数: 0 h-index: 0机构: Henry Ford Hosp, Detroit, MI USA Queen Elizabeth Hosp TQEH, Woodville South, AustraliaRichardson, Gary论文数: 0 引用数: 0 h-index: 0机构: Cabrini Hosp Malvern, Malvern, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaUnderhill, Craig论文数: 0 引用数: 0 h-index: 0机构: Border Med Oncol, Albury Wodonga, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaGanju, Vinod论文数: 0 引用数: 0 h-index: 0机构: Peninsula Oncol Ctr, Victoria, Australia Queen Elizabeth Hosp TQEH, Woodville South, AustraliaLee, Keun-Wook论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Bundang, Seoul Natl Univ, Coll Med, Seongnam, South Korea Queen Elizabeth Hosp TQEH, Woodville South, AustraliaHuh, Seok Jae论文数: 0 引用数: 0 h-index: 0机构: Dong A Univ Hosp, Seogu, South Korea Queen Elizabeth Hosp TQEH, Woodville South, AustraliaKim, Sang-We论文数: 0 引用数: 0 h-index: 0机构: Asan Med Ctr, Seoul, South Korea Queen Elizabeth Hosp TQEH, Woodville South, AustraliaYang, Chih-Hsin论文数: 0 引用数: 0 h-index: 0机构: Natl Taiwan Univ Hosp, Taipei, Taiwan Queen Elizabeth Hosp TQEH, Woodville South, AustraliaChen, Yuh-Min论文数: 0 引用数: 0 h-index: 0机构: Taichung Vet Gen Hosp, Dept Chest Med, Taipei, Taiwan Queen Elizabeth Hosp TQEH, Woodville South, AustraliaXiang, Ziyong论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, AustraliaShi, Zhe论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, AustraliaWang, Yaolin论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, AustraliaZhang, Ling论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp TQEH, Woodville South, AustraliaMillward, Michael论文数: 0 引用数: 0 h-index: 0机构: Norton Canc Inst, Louisville, KY USA Linear Clin Res Ltd, Nedlands, Australia Queen Elizabeth Hosp TQEH, Woodville South, Australia
- [33] First-in-human phase I trial of the PI3Kb-selective inhibitor SAR260301 in patients with advanced solid tumors (NCT01673737).JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Bedard, Philippe L.论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaDavies, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaKopetz, Scott论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaFlaherty, Keith T.论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaShapiro, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaLuke, Jason John论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaSpreafico, Anna论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaWu, Bin论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaGomez, Corinne论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaCartot-Cotton, Sylvaine论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaMazuir, Florent论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaMicallef, Sandrine论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaDemers, Brigitte论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, CanadaJuric, Dejan论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Toronto, ON, Canada
- [34] First-in-Human Phase I Study of GSK2126458, an Oral Pan-Class I Phosphatidylinositol-3-Kinase Inhibitor, in Patients with Advanced Solid Tumor MalignanciesCLINICAL CANCER RESEARCH, 2016, 22 (08) : 1932 - 1939Munster, Pamela论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAAggarwal, Rahul论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAHong, David论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USASchellens, Jan H. M.论文数: 0 引用数: 0 h-index: 0机构: Netherlands Canc Inst, Amsterdam, Netherlands Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAvan der Noll, Ruud论文数: 0 引用数: 0 h-index: 0机构: Netherlands Canc Inst, Amsterdam, Netherlands Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USASpecht, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Fred Hutchinson Canc Res Ctr, 1124 Columbia St, Seattle, WA 98104 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAWitteveen, Petronella O.论文数: 0 引用数: 0 h-index: 0机构: Univ Utrecht, Ctr Canc, NL-3508 TC Utrecht, Netherlands Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAWerner, Theresa L.论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Huntsman Canc Inst, Salt Lake City, UT USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USADees, E. Claire论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comprehens Canc Ctr, Chapel Hill, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USABergsland, Emily论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USA论文数: 引用数: h-index:机构:Kleha, Joseph F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USADurante, Michael论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAAdams, Laurel论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USASmith, Deborah A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USALampkin, Thomas A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAMorris, Shannon R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USAKurzrock, Razelle论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Calif San Francisco, 1600 Divisadero St,Rm A719 Box 1711, San Francisco, CA 94143 USA
- [35] First-in-human (FIH) phase I study of GST-HG161, a potent and highly selective c-met inhibitor, in patients with advanced solid tumor.JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (15)Li, Jin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaGuo, Ye论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXue, Junli论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaWu, Wenqiang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChen, Shikui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaTang, Yanan论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXu, Xiongbin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaLi, Gang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaHu, Lihong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaLin, Yunfei论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaShen, Liang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXia, Yuanfeng论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChan, Chi-Chung论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaWang, Zhouchong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaNi, Dawen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaDing, Charles论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChen, Shuhui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R China
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- [37] Trial in progress: A phase 1, first-in-human, open-label, multicenter, dose-escalation and dose-expansion study of ASP3082 in patients with previously treated advanced solid tumors and KRAS G12D mutations.JOURNAL OF CLINICAL ONCOLOGY, 2023, 41 : TPS764 - TPS764Tolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAPark, Wungki论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAWang, Judy S.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USASpira, Alexander I.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USALee, Ho-Jin论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAGill, Stanley论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USALoRusso, Patricia论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAHerzberg, Benjamin论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAGoldman, Jonathan W.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAMorgensztern, Daniel论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USABerlin, Jordan论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAKasi, Anup论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAFujii, Hisaki论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USAPelster, Meredith论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USA
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