CONDENSED HETEROCYCLIC LACTAMS .2. SYNTHESIS OF NEW 4-ARYLQUINOLIN-2(1H)-ONE DERIVATIVES

被引：0
|
作者：
HAZAI, L
DEAK, G
TOTH, G
SOHAR, P
TAMAS, J
GYORGY, L
机构：
[1] TECH UNIV BUDAPEST,INST GEN & ANALYT CHEM,H-1111 BUDAPEST,HUNGARY
[2] EGIS PHARMACEUT,DEPT SPECTROSCOP,H-1475 BUDAPEST,HUNGARY
[3] HUNGARIAN ACAD SCI,INST EXPTL MED,H-1450 BUDAPEST,HUNGARY
[4] HUNGARIAN ACAD SCI,CENT RES INST CHEM,H-1525 BUDAPEST,HUNGARY
来源：
ACTA CHIMICA HUNGARICA-MODELS IN CHEMISTRY | 1992年 / 129卷 / 02期
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Catalytic hydrogenation of the nitro group of 4-(4-nitrophenyl)quinolin-2(1H)-one (1) gave, without saturation of the C-3 - C-4 double bond, a new representative of 4-arylquinolin-2(1H)-ones: the 4-(4-aminophenyl) derivative 3. The use of this compound as a starting material made possible the syntheses of potentially CNS active 4-alkylaminoacylamino-substituted 4-arylquinolin-2(1H)-ones (6a-d) and related compounds (6e-j).
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页码：269 / 275
页数：7
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