ANGIOTENSIN-II ANTAGONISTS WHICH EXHIBIT EQUAL BINDING AFFINITIES FOR BOTH THE AT1 AND AT2 RECEPTOR SUBTYPES

被引:0
|
作者
SANTELLA, JB [1 ]
ENSINGER, CL [1 ]
VANATTEN, MK [1 ]
CARINI, DJ [1 ]
WEXLER, RR [1 ]
CHIU, AT [1 ]
MCCALL, DE [1 ]
WONG, PC [1 ]
TIMMERMANS, PBMWM [1 ]
DUNCIA, JV [1 ]
机构
[1] DUPONT MERCK PHARMACEUT CO,WILMINGTON,DE 19880
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:199 / MEDI
相关论文
共 50 条
  • [21] Ontogeny and regulation of cardiac angiotensin II receptor subtypes (AT1 and AT2) in developing sheep.
    Segar, JL
    Bedell, KA
    Mathews, MS
    Petershack, JE
    Robillard, JE
    PEDIATRIC RESEARCH, 1996, 39 (04) : 205 - 205
  • [22] Antagonists of the AT1 receptor for angiotensin II
    Kawecka-Jaszcz, Kalina
    Czarnecka, Danuta
    Wojciechowska, Wiktoria
    ARTERIAL HYPERTENSION, 2006, 10 : A1 - A15
  • [23] POTENT IMIDAZOPYRIDINE ANGIOTENSIN-II ANTAGONISTS WITH BALANCED AFFINITY TO AT(1) AND AT(2) RECEPTOR SUBTYPES
    KIM, D
    MANTLO, NB
    ONDEYKA, D
    CHANG, RSL
    KIVLIGHN, SD
    SIEGL, PKS
    GREENLEE, WJ
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 207 : 208 - MEDI
  • [24] DEVELOPMENT OF ANGIOTENSIN-II ANTAGONISTS WITH EQUIPOTENT AFFINITY FOR HUMAN AT(1) AND AT(2) RECEPTOR SUBTYPES
    GLINKA, TW
    DELASZLO, SE
    SIEGL, PKS
    CHANG, RS
    KIVLIGHN, SD
    SCHORN, TS
    FAUST, KA
    CHEN, TB
    ZINGARO, GJ
    LOTTI, VJ
    GREENLEE, WJ
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1994, 4 (19) : 2337 - 2342
  • [25] EXP597, A NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONIST WITH HIGH AFFINITIES FOR THE ANGIOTENSIN AT(1) AND AT(2) RECEPTOR SUBTYPES
    WONG, PC
    DUNCIA, JV
    SANTELLA, JB
    SMITH, RD
    WEXLER, RR
    TIMMERMANS, PBMWM
    CHIU, AT
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1994, 260 (2-3) : 261 - 264
  • [26] Balanced affinity AT1/AT2 receptor nonpeptide binding site determinants on the AT1 angiotensin receptor
    Clarke, D
    Sothinathan, R
    Speth, RC
    Sandberg, K
    INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE, 1998, 2 (02) : 197 - 201
  • [27] ANGIOTENSIN-II RECEPTOR SUBTYPES - SELECTIVE ANTAGONISTS AND FUNCTIONAL CORRELATES
    TIMMERMANS, PBMWM
    SMITH, RD
    EUROPEAN HEART JOURNAL, 1994, 15 : 79 - 87
  • [28] BALANCED ANGIOTENSIN-II RECEPTOR ANTAGONISTS .1. THE EFFECTS OF BIPHENYL ORTHO SUBSTITUTION ON AT(1)/AT(2) AFFINITIES
    QUAN, ML
    OLSON, RE
    CARINI, DJ
    ELLIS, CD
    HILLYER, GL
    LALKA, GK
    LIU, J
    VANATTEN, MK
    CHIU, AT
    WONG, PC
    WEXLER, RR
    TIMMERMANS, PBMWM
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1994, 4 (16) : 2011 - 2016
  • [29] Increased Angiotensin II AT1 receptor mRNA and binding in spleen and lung of AT2 receptor gene disrupted mice
    Pavel, Jaroslav
    Terron, Jose A.
    Benicky, Julius
    Falcon-Neri, Alicia
    Rachakonda, Amita
    Inagami, Tadashi
    Saavedra, Juan M.
    REGULATORY PEPTIDES, 2009, 158 (1-3) : 156 - 166
  • [30] SYNTHESIS OF N-ALKYL-1,2,4-OXADIAZINONES AS ANGIOTENSIN-II (AT1) RECEPTOR ANTAGONISTS
    WELLER, HN
    MILLER, AV
    DICKINSON, KEJ
    HEDBERG, SA
    DELANEY, CL
    SERAFINO, RP
    MORELAND, S
    HETEROCYCLES, 1993, 36 (05) : 1027 - 1038