ANGIOTENSIN-II ANTAGONISTS WHICH EXHIBIT EQUAL BINDING AFFINITIES FOR BOTH THE AT1 AND AT2 RECEPTOR SUBTYPES

被引:0
|
作者
SANTELLA, JB [1 ]
ENSINGER, CL [1 ]
VANATTEN, MK [1 ]
CARINI, DJ [1 ]
WEXLER, RR [1 ]
CHIU, AT [1 ]
MCCALL, DE [1 ]
WONG, PC [1 ]
TIMMERMANS, PBMWM [1 ]
DUNCIA, JV [1 ]
机构
[1] DUPONT MERCK PHARMACEUT CO,WILMINGTON,DE 19880
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:199 / MEDI
相关论文
共 50 条
  • [1] BALANCED AT1/AT2 ANGIOTENSIN-II RECEPTOR ANTAGONISTS
    QUAN, ML
    OLSON, RE
    CARINI, DJ
    ELLIS, CD
    LALKA, GK
    LIU, J
    VANATTEN, MK
    WEXLER, RR
    CHIU, AT
    WONG, PC
    TIMMERMANS, PBMWM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 207 : 201 - MEDI
  • [2] TRIAZOLINONE SULFONAMIDES WITH HIGH-AFFINITY FOR BOTH THE AT1 AND THE AT2 SUBTYPES OF THE ANGIOTENSIN-II RECEPTOR
    CHANG, LL
    ASHTON, WT
    FLANAGAN, KL
    CHANG, RSL
    LOTTI, VJ
    GREENLEE, WJ
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 207 : 13 - MEDI
  • [3] NONPEPTIDE ANGIOTENSIN-II ANTAGONISTS WITH AFFINITY FOR AT1 AND AT2 RECEPTORS
    OLSON, RE
    LIN, J
    LALKA, GK
    DUNCIO, JV
    WEXLER, RR
    CHIU, AT
    MCCALL, DE
    WONG, P
    TIMMERMANS, PBMWM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1993, 206 : 77 - MEDI
  • [4] CHARACTERIZATION AND DEVELOPMENT OF ANGIOTENSIN-II RECEPTOR SUBTYPES (AT1 AND AT2) IN RAT-BRAIN
    TSUTSUMI, K
    SAAVEDRA, JM
    AMERICAN JOURNAL OF PHYSIOLOGY, 1991, 261 (01): : R209 - R216
  • [5] AMPHIBIAN MYOCARDIAL ANGIOTENSIN-II RECEPTORS ARE DISTINCT FROM MAMMALIAN AT1 AND AT2 RECEPTOR SUBTYPES
    SANDBERG, K
    JI, H
    MILLAN, MA
    CATT, KJ
    FEBS LETTERS, 1991, 284 (02) : 281 - 284
  • [6] DIFFERENTIAL DISTRIBUTION OF AT1 AND AT2 ANGIOTENSIN-II RECEPTOR SUBTYPES IN THE RAT-BRAIN DURING DEVELOPMENT
    MILLAN, MA
    JACOBOWITZ, DM
    AGUILERA, G
    CATT, KJ
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1991, 88 (24) : 11440 - 11444
  • [7] Angiotensin II receptor subtypes AT1 and AT2 are down-regulated by angiotensin II through AT1 receptor by different mechanisms
    Ouali, R
    Berthelon, MC
    Begeot, M
    Saez, JM
    ENDOCRINOLOGY, 1997, 138 (02) : 725 - 733
  • [8] Effects of AT1 and AT2 angiotensin receptor antagonists in angiotensin II-infused rats
    Li, JS
    Touyz, RM
    Schiffrin, EL
    HYPERTENSION, 1998, 31 (01) : 487 - 492
  • [9] RADIOIODINATED NONPEPTIDE, ANGIOTENSIN-II AT1 RECEPTOR ANTAGONISTS
    BURNS, HD
    BRENNER, NJ
    GIBSON, RE
    BEAUCHAMP, HT
    CHANG, RS
    FIORAVANTI, C
    NAYLOR, EM
    JOURNAL OF NUCLEAR MEDICINE, 1994, 35 (05) : P246 - P246
  • [10] ANGIOTENSIN-II RECEPTOR ANTAGONISTS AND RECEPTOR SUBTYPES
    WONG, PC
    CHIU, AT
    DUNCIA, JV
    HERBLIN, WF
    SMITH, RD
    TIMMERMANS, PBMWM
    TRENDS IN ENDOCRINOLOGY AND METABOLISM, 1992, 3 (06): : 211 - 217