ASYMMETRIC-SYNTHESIS OF (3S)-2,3,4,5-TETRAHYDROPYRIDAZINE-3-CARBOXYLIC ACID

被引：43

作者：

ASPINALL, IH

COWLEY, PM

MITCHELL, G

STOODLEY, RJ

机构：

[1] UMIST,DEPT CHEM,POB 88,MANCHESTER M60 1QD,ENGLAND

[2] ZENECA AGROCHEM,JEALOTTS HILL RES STN,BRACKNELL RG12 6EY,BERKS,ENGLAND

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1993年 / 15期

关键词：

D O I：

10.1039/c39930001179

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The title compound 1a is prepared by a two-step sequence from the cycloadduct 5d, derived from di(tert-butyl) azodicarboxylate and the diene 4b by a hetero Diels-Alder reaction.

引用

页码：1179 / 1180

页数：2

共 50 条

[21] ASYMMETRIC-SYNTHESIS VIA ACETAL TEMPLATES .14. PREPARATION OF ENANTIOMERICALLY PURE (3S,4S)-STATINE AND (3S,4R)-STATINE DERIVATIVES
ANDREW, RG
CONROW, RE
ELLIOTT, JD
JOHNSON, WS
RAMEZANI, S
TETRAHEDRON LETTERS, 1987, 28 (52) : 6535 - 6538
[22] Asymmetric synthesis of (2R,3S)-3-hydroxypipecolic acid δ-lactam derivatives
Koulocheri, SD
Magiatis, P
Skaltsounis, AL
Haroutounian, SA
TETRAHEDRON, 2002, 58 (33) : 6665 - 6671
[23] (2S,3S)-3-(4-Chlorophenyl)-8-methyltropane2-carboxylic acid
Chen, Zheng-Ping
Wang, Song-Pei
Li, Xiao-Min
Tang, Jie
Lin, Jian-Guo
ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2008, 64 : O1732 - U1701
[24] ASYMMETRIC-SYNTHESIS OF 3S,4R-DIHYDROXYPYRROLIDINES BY REGIOSELECTIVE AND STEREOSELECTIVE HYDROXYLATION OF 4-OXOPROLINE ENOLATE
BLANCO, MJ
SARDINA, FJ
TETRAHEDRON LETTERS, 1994, 35 (45) : 8493 - 8496
[25] AN EFFICIENT ASYMMETRIC-SYNTHESIS OF (R)-3-AMINO-2,3,4,5-TETRAHYDRO-1H-[1]BENZAZEPIN-2-ONE
ARMSTRONG, JD
ENG, KK
KELLER, JL
PURICK, RM
HARTNER, FW
CHOI, WB
ASKIN, D
VOLANTE, RP
TETRAHEDRON LETTERS, 1994, 35 (20) : 3239 - 3242
[26] ASYMMETRIC-SYNTHESIS OF ORGANOELEMENTAL ANALOGS OF NATURAL COMPOUNDS .7. (2R,3S)-2-AMINO-3-HYDROXY-5-PHOSPHONOVALERIC ACID
SOLOSHONOK, VA
SVISTUNOVA, NY
KUKHAR, VP
GUDIMA, AO
KUZMINA, NA
BELOKON, YN
BULLETIN OF THE RUSSIAN ACADEMY OF SCIENCES-DIVISION OF CHEMICAL SCIENCE, 1992, 41 (05): : 922 - 925
[27] An asymmetric dihydroxylation route to (2S,3S)-3-hydroxypipecolic acid
Bodas, MS
Kumar, P
TETRAHEDRON LETTERS, 2004, 45 (46) : 8461 - 8463
[28] A SUCCINCT ASYMMETRIC-SYNTHESIS OF (2S,3R)-2-METHYL-3-AMINOPENTANOIC ACID HYDROCHLORIDE
DAVIES, SG
ICHIHARA, O
WALTERS, IAS
SYNLETT, 1994, (02) : 117 - 118
[29] Asymmetric synthesis of novel highly sterically constrained (2S,3S)-3-methyl-3-trifluoromethyl- and (2S,3S,4R)-3-trifluoromethyl-4-methylpyroglutamic acids
Soloshonok, VA
Cai, CZ
Hruby, VJ
TETRAHEDRON, 1999, 55 (41) : 12045 - 12058
[30] The first asymmetric synthesis of (2S,3S,4R)-3-amino-2-hydroxymethyl-4-hydroxypyrrolidine
Curtis, KL
Fawcett, J
Handa, S
TETRAHEDRON LETTERS, 2005, 46 (32) : 5297 - 5300

← 1 2 3 4 5 →