RAPAMYCIN AND FK506 BINDING-PROTEINS (IMMUNOPHILINS)

被引:148
|
作者
FRETZ, H
ALBERS, MW
GALAT, A
STANDAERT, RF
LANE, WS
BURAKOFF, SJ
BIERER, BE
SCHREIBER, SL
机构
[1] HARVARD UNIV,DEPT CHEM,CAMBRIDGE,MA 02138
[2] HARVARD UNIV,SCH MED,DANA FARBER CANC INST,DIV PEDIAT ONCOL,BOSTON,MA 02115
关键词
D O I
10.1021/ja00004a051
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:1409 / 1411
页数:3
相关论文
共 50 条
  • [21] Analogous conformations of both binding and effector regions in cyclosporin A, FK506 and rapamycin
    Denesyuk, AI
    Denessiouk, KA
    Zav'yalov, VP
    Lundell, J
    Korpela, T
    COMPUTERS & CHEMISTRY, 1998, 22 (04): : 339 - 344
  • [22] Structure of the human 25 kDa FK506 binding protein complexed with rapamycin
    Liang, J
    Hung, DT
    Schreiber, SL
    Clardy, J
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1996, 118 (05) : 1231 - 1232
  • [23] Evaluation of Synthetic FK506 Analogues as Ligands for the FK506-Binding Proteins 51 and 52
    Gopalakrishnan, Ranganath
    Kozany, Christian
    Gaali, Steffen
    Kress, Christoph
    Hoogeland, Bastiaan
    Bracher, Andreas
    Hausch, Felix
    JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (09) : 4114 - 4122
  • [24] Comparison of acute rapamycin nephrotoxicity with cyclosporine and FK506
    Andoh, TF
    Burdmann, EA
    Fransechini, N
    Houghton, DC
    Bennett, WM
    KIDNEY INTERNATIONAL, 1996, 50 (04) : 1110 - 1117
  • [25] MODES OF ACTION OF FK506, CYCLOSPORINE-A, AND RAPAMYCIN
    MORRIS, R
    TRANSPLANTATION PROCEEDINGS, 1994, 26 (06) : 3272 - 3275
  • [26] Effect of rapamycin and FK506 on mesangial cell proliferation
    Wang, W
    Chan, YH
    Lee, W
    Chan, L
    TRANSPLANTATION PROCEEDINGS, 2001, 33 (1-2) : 1036 - 1037
  • [27] The antimalarial action of FK506 and rapamycin: evidence for a direct effect on FK506-binding protein PfFKBP35
    Monaghan, Paul
    Leneghan, Darren B.
    Shaw, Wesley
    Bell, Angus
    PARASITOLOGY, 2017, 144 (07) : 869 - 876
  • [28] Large FK506-Binding Proteins Shape the Pharmacology of Rapamycin
    Maerz, Andreas M.
    Fabian, Anne-Katrin
    Kozany, Christian
    Bracher, Andreas
    Hausch, Felix
    MOLECULAR AND CELLULAR BIOLOGY, 2013, 33 (07) : 1357 - 1367
  • [29] COMPARATIVE X-RAY STRUCTURES OF THE MAJOR BINDING-PROTEIN FOR THE IMMUNOSUPPRESSANT FK506 (TACROLIMUS) IN UNLIGANDED FORM AND IN COMPLEX WITH FK506 AND RAPAMYCIN
    WILSON, KP
    YAMASHITA, MM
    SINTCHAK, MD
    ROTSTEIN, SH
    MURCKO, MA
    BOGER, J
    THOMSON, JA
    FITZGIBBON, MJ
    BLACK, JR
    NAVIA, MA
    ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY, 1995, 51 : 511 - 521
  • [30] HEPATOTROPHIC PROPERTIES IN DOGS OF HUMAN FKBP, THE BINDING-PROTEIN FOR FK506 AND RAPAMYCIN
    STARZL, TE
    SCHREIBER, SL
    ALBERS, MW
    PORTER, KA
    FOGLIENI, CS
    FRANCAVILLA, A
    TRANSPLANTATION, 1991, 52 (04) : 751 - 753