SYNTHESIS OF THIAZOLE AND SELENAZOLE DERIVATIVES WITH AFFINITY FOR THE ODORANT-BINDING PROTEIN

被引：7

作者：

NAPOLITANO, E

PELOSI, P

机构：

[1] UNIV PISA,IST IND AGR,VIA S MICHELE 4,I-56124 PISA,ITALY

[2] UNIV PISA,DIPARTIMENTO CHIM BIOORGAN,I-56100 PISA,ITALY

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1992年 / 2卷 / 12期

关键词：

D O I：

10.1016/S0960-894X(00)80439-4

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Three new ligands for odorant-binding proteins (OBPs) have been prepared, to be used in protein structure studies: the photoaffinity label 2-azido-4-butyl-5-propylthiazole, the NMR probe 2-trifluoromethyl-4-butyl-5-propylthiazole and the X-ray probe 2-amino-4-butyl-5-propylselenazole. All three compounds bind the bovine OBP with dissociation constants in the micromolar range.

引用

页码：1603 / 1606

页数：4

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