BLOCKADE OF INVIVO BINDING OF I-125-LABELED 3-IODOBENZAMIDE (IBZM) TO DOPAMINE-RECEPTORS BY D2 ANTAGONIST AND AGONIST

被引:12
|
作者
SINGHANIYOM, W
TSAI, YF
BRUCKE, T
MCLELLAN, CA
COHEN, RM
KUNG, HF
CHIUEH, CC
机构
[1] NIMH, CEREBRAL METAB LAB,CLIN BRAIN IMAGING SECT, BLDG 10,RM 2D-52, BETHESDA, MD 20892 USA
[2] UNIV PENN, DEPT RADIOL, PHILADELPHIA, PA 19104 USA
关键词
D O I
10.1016/0006-8993(88)90186-2
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:393 / 396
页数:4
相关论文
共 50 条
  • [21] ERGOVALINE BINDING AND ACTIVATION OF D2 DOPAMINE-RECEPTORS IN GH(4)ZR(7) CELLS
    LARSON, BT
    SAMFORD, MD
    CAMDEN, JM
    PIPER, EL
    KERLEY, MS
    PATERSON, JA
    TURNER, JT
    JOURNAL OF ANIMAL SCIENCE, 1995, 73 (05) : 1396 - 1400
  • [22] D2 DOPAMINE-RECEPTORS IN RAT STRIATUM ARE HOMOGENEOUS AS REVEALED BY LIGAND-BINDING STUDIES
    LEONARD, MN
    HALLIDAY, CA
    MARRIOTT, AS
    STRANGE, PG
    BIOCHEMICAL PHARMACOLOGY, 1988, 37 (22) : 4335 - 4339
  • [23] Striatal dopamine D2/3 receptors in medication-naive schizophrenia: an [123I] IBZM SPECT study
    Chen, Kao Chin
    Yang, Yen Kuang
    Howes, Oliver D.
    Lee, I. Hui
    Yeh, Tzung Lieh
    Chiu, Nan Tsing
    Chen, Po See
    David, Anthony S.
    Bramon, Elvira
    PSYCHOLOGICAL MEDICINE, 2022, 52 (14) : 3251 - 3259
  • [24] Agonist action at D2(long) dopamine receptors:: ligand binding and functional assays
    Gardner, B
    Strange, PG
    BRITISH JOURNAL OF PHARMACOLOGY, 1998, 124 (05) : 978 - 984
  • [25] Rotigotine is a potent agonist at dopamine D1 receptors as well as at dopamine D2 and D3 receptors
    Wood, Martyn
    Dubois, Vanessa
    Scheller, Dieter
    Gillard, Michel
    BRITISH JOURNAL OF PHARMACOLOGY, 2015, 172 (04) : 1124 - 1135
  • [26] STIMULANT-CONDITIONED LOCOMOTION IS NOT AFFECTED BY BLOCKADE OF D1 AND OR D2 DOPAMINE-RECEPTORS DURING CONDITIONING
    MARTINIVERSON, MT
    MCMANUS, DJ
    BRAIN RESEARCH, 1990, 521 (1-2) : 175 - 184
  • [27] [H-3] SPIPERONE BINDS SELECTIVELY TO RAT STRIATAL D2 DOPAMINE-RECEPTORS INVIVO - A KINETIC AND PHARMACOLOGICAL ANALYSIS
    LESLIE, CA
    BENNETT, JP
    BRAIN RESEARCH, 1987, 407 (02) : 253 - 262
  • [28] Evaluation of the distribution of dopamine D2 receptors with I-123 IBZM SPECT in unilateral dystonias.
    Lang, O
    Stejskal, L
    Ruzicka, E
    Holy, R
    Balon, HR
    JOURNAL OF NUCLEAR MEDICINE, 2003, 44 (05) : 234P - 234P
  • [29] I-chloroscoulerine mesylate -: Antipsychotic dopamine D1 agonist/D2 antagonist
    Li, Jianfeng
    Jin, Guozhang
    Shen, Jingshan
    Shanghai, Ruyun A.
    DRUGS OF THE FUTURE, 2006, 31 (05) : 379 - 384
  • [30] QUANTITATIVE AUTORADIOGRAPHIC DEMONSTRATION OF HIGH AND LOW AFFINITY AGONIST BINDING OF D-2 DOPAMINE-RECEPTORS
    DAWSON, TM
    GEHLERT, DR
    WAMSLEY, JK
    CLINICAL RESEARCH, 1985, 33 (02): : A282 - A282