SYNTHESIS AND HERBICIDAL ACTIVITY OF PHENOXYPROPIONIC ACID-DERIVATIVES WITH IMIDAZO[1,2-A]PYRIDINE MOIETY

被引:6
|
作者
OHTA, K
MINAMI, K
YOSHIKAWA, H
ISHIDA, Y
机构
[1] Agricultural Research Laboratories, Agro Division, Takeda Chemical Industries Ltd., Tsukuba, Ibaraki 300-42
关键词
D O I
10.1271/bbb.57.1844
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
Phenoxypropionic acid derivatives (Ia-s) with an imidazo[1,2-a]pyridine moiety were synthesized and their herbicidal activities were examined. The activities were affected dramatically by the substituents on the imidazo[1,2-a]pyridine ring, and good substituents to enhance the herbicidal activity were a cyano group at the 3-position and a chlorine atom at the 6-position. Among the compounds, n-propyl 2-[4-(6-chloro-3-cyano-2-imidazo[1,2-a]pyridinvloxy)phenoxy]propionate(Iq) was most active against gramineous weeds and the activity was comparable to that of the commercial herbicide fluazifop-butyl.
引用
收藏
页码:1844 / 1848
页数:5
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