1,3-ASYMMETRIC INDUCTION - HIGHLY ENANTIOSELECTIVE SYNTHESIS OF ALPHA-AMINO-ACIDS VIA 2,5-TRANS DISUBSTITUTED IMIDAZOLIDIN-4-ONES

被引：17

作者：

AMOROSO, R ^{[1
]}

CARDILLO, G ^{[1
]}

TOMASINI, C ^{[1
]}

机构：

[1] UNIV BOLOGNA,CTR STUDIO FIS MACROMOLEC,DIPARTIMENTO CHIM G CIAMICIAN,I-40126 BOLOGNA,ITALY

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 17期

关键词：

D O I：

10.1016/0040-4039(91)85016-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2,5-Trans imidazolidin-4-ones have been obtained from mercury promoted cyclisation of unsaturated amidals containing a stereogenic centre. A new enantioselective synthesis of alpha-amino acids has been devised.

引用

页码：1971 / 1974

页数：4

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