COMPARISON OF LOCATION AND BINDING FOR THE POSITIVELY CHARGED 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL ANTAGONIST AMLODIPINE WITH UNCHARGED DRUGS OF THIS CLASS IN CARDIAC MEMBRANES

被引：0
|
作者：
MASON, RP
CAMPBELL, SF
WANG, SD
HERBETTE, LG
机构：
[1] UNIV CONNECTICUT,CTR HLTH,CTR BIOMOLEC STRUCT ANAL,FARMINGTON,CT 06032
[2] UNIV CONNECTICUT,CTR HLTH,DEPT BIOCHEM,FARMINGTON,CT 06032
[3] PFIZER LTD,DEPT DISCOVERY CHEM,SANDWICH CT13 9NJ,KENT,ENGLAND
[4] UNIV CONNECTICUT,CTR HLTH,DEPT RADIOL,FARMINGTON,CT 06032
[5] UNIV CONNECTICUT,CTR HLTH,DEPT MED,FARMINGTON,CT 06032
来源：
MOLECULAR PHARMACOLOGY | 1989年 / 36卷 / 04期
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：634 / 640
页数：7
相关论文
共 50 条
  • [41] Synthesis and calcium channel antagonist activity of 1,4-dihydropyridine derivatives containing 4-nitroimidazolyl substituents
    Shafiee, A
    Rastkary, N
    Jorjani, M
    ARZNEIMITTELFORSCHUNG-DRUG RESEARCH, 2002, 52 (07): : 537 - 542
  • [42] IDENTIFICATION OF A NOVEL 1,4-DIHYDROPYRIDINE-BINDING AND PHENYLALKYLAMINE-BINDING POLYPEPTIDE IN CALCIUM-CHANNEL PREPARATIONS
    VAGHY, PL
    STRIESSNIG, J
    MIWA, K
    KNAUS, HG
    ITAGAKI, K
    MCKENNA, E
    GLOSSMANN, H
    SCHWARTZ, A
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1987, 262 (29) : 14337 - 14342
  • [43] PROBING MEMBRANE BILAYER INTERACTIONS OF 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL BLOCKERS - IMPLICATIONS FOR AGING AND ALZHEIMERS-DISEASE
    MASON, RP
    CALCIUM HYPOTHESIS OF AGING AND DEMENTIA, 1994, 747 : 125 - 139
  • [44] PHOTOAFFINITY-LABELING OF A 33-35,000 DALTON PROTEIN IN CARDIAC, SKELETAL AND SMOOTH-MUSCLE MEMBRANES USING A NEW I-125 LABELED 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL ANTAGONIST
    SARMIENTO, JG
    EPSTEIN, PM
    ROWE, WA
    CHESTER, DW
    SMILOWITZ, H
    WEHINGER, E
    JANIS, RA
    LIFE SCIENCES, 1986, 39 (25) : 2401 - 2409
  • [45] 1,4-DIHYDROPYRIDINE CA-2+ CHANNEL ANTAGONISTS AND ACTIVATORS - A COMPARISON OF BINDING CHARACTERISTICS WITH PHARMACOLOGY
    JANIS, RA
    TRIGGLE, DJ
    DRUG DEVELOPMENT RESEARCH, 1984, 4 (03) : 257 - 274
  • [46] Synthesis and calcium channel antagonist activity of novel 1,4-dihydropyridine derivatives possessing 4-pyrone moieties
    Aziz Shahrisa
    Ramin Miri
    Somayeh Esmati
    Mahnaz Saraei
    Ahmad Reza Mehdipour
    Maryam Sharifi
    Medicinal Chemistry Research, 2012, 21 : 284 - 292
  • [47] Synthesis and calcium channel antagonist activity of novel 1,4-dihydropyridine derivatives possessing 4-pyrone moieties
    Shahrisa, Aziz
    Miri, Ramin
    Esmati, Somayeh
    Saraei, Mahnaz
    Mehdipour, Ahmad Reza
    Sharifi, Maryam
    MEDICINAL CHEMISTRY RESEARCH, 2012, 21 (03) : 284 - 292
  • [48] REGULATION OF THE NUMBER OF ALPHA-BUNGAROTOXIN BINDING-SITES IN CULTURED CHICK MYOTUBES BY A 1,4 DIHYDROPYRIDINE CALCIUM-CHANNEL ANTAGONIST
    SMILOWITZ, H
    SMART, E
    BOWIK, C
    CHANG, RJ
    JOURNAL OF NEUROSCIENCE RESEARCH, 1988, 19 (03) : 321 - 325
  • [49] EFFECTS OF ANTI-CALCIUM CHANNEL ALPHA-2-SUBUNIT ANTIBODIES ON CALCIUM FLUX AND 1,4-DIHYDROPYRIDINE BINDING
    KOWALSKI, MT
    GEORGE, PR
    HARRISON, TM
    WRAY, DW
    NORMAN, RI
    BIOCHEMICAL SOCIETY TRANSACTIONS, 1990, 18 (05) : 890 - 890
  • [50] CARDIOVASCULAR EFFECTS OF OPC-13340, A POTENT, LONG-ACTING 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL BLOCKER, IN DOGS
    MORI, T
    NAKAYAMA, N
    OHURA, M
    IKEZONO, K
    KINOSHITA, S
    KAMATA, M
    HOSOKAWA, T
    YAMASHITA, S
    YABUUCHI, Y
    ARCHIVES INTERNATIONALES DE PHARMACODYNAMIE ET DE THERAPIE, 1993, 321 : 41 - 56
12345