THE 3,4-DIMETHOXYBENZYL MOIETY AS A NEW N-PROTECTING GROUP OF 1,2-THIAZETIDINE 1,1-DIOXIDES

被引：20

作者：

GRUNDERKLOTZ, E

EHRHARDT, JD

机构：

[1] Laboratoire de Pharmacologie Cardiovasculaire et Rénale, associé au CNRS, Université Louis Pasteur, 6700 Strasbourg

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(00)74875-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The 3,4-dimethoxybenzyl group was used to N-protect 3,4-diphenyl 1, 2-thiazetidine 1, 1-dioxide derivatives. It is smoothly eliminated by 2,3-dichloro 5,6-dicyanobenzoquinone (DDQ), the yield depending on the substituents of the 3-phenyl ring.

引用

页码：751 / 752

页数：2

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