NOVEL ORALLY ACTIVE INHIBITORS OF PASSIVE CUTANEOUS ANAPHYLAXIS IN RATS - N-[2-(4-PYRIDINYL)-4-PYRIMIDINYL]UREAS AND DIALKYL[[[2-(4-PYRIDINYL)-4-PYRIMIDINYL]AMINO]METHYLENE]MALONATES

被引：13

作者：

LESHER, GY

SINGH, B

MIELENS, ZE

机构：

[1] STERLING WINTHROP RES INST,DEPT MED CHEM,RENSSELAER,NY 12144

[2] STERLING WINTHROP RES INST,DEPT OBSTET & GYNECOL,RENSSELAER,NY 12144

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1982年 / 25卷 / 07期

关键词：

D O I：

10.1021/jm00349a014

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：837 / 842

页数：6

共 50 条

[21] Metal-Metal Quadruple Bonds (M = Mo or W) Supported by 4-[2-(4-Pyridinyl)ethenyl] Benzoates and their Complexes with Tris(pentafluorophenyl)boron
Chisholm, Malcolm H.
Ziehm, Christopher J.
INORGANIC CHEMISTRY, 2015, 54 (23) : 11168 - 11173
[22] Characterization of 2-[[4-Fluoro-3-(trifluoromethyl)phenyl]amino]-4-(4-pyridinyl)-5-thiazolemethanol (JNJ-1930942), a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Receptor
Dinklo, Theo
Shaban, Hamdy
Thuring, Jan Willem
Lavreysen, Hilde
Stevens, Karen E.
Zheng, Lijun
Mackie, Claire
Grantham, Christopher
Vandenberk, Ine
Meulders, Greet
Peeters, Luc
Verachtert, Hanne
De Prins, Erik
Lesage, Anne S. J.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2011, 336 (02): : 560 - 574
[23] Potent and selective ET-A antagonists.: 2.: Discovery and evaluation of potent and water soluble N-(6-(2-(aryloxy)ethoxy)-4-pyrimidinyl)sulfonamide derivatives
Morimoto, H
Ohashi, N
Shimadzu, H
Kushiyama, E
Kawanishi, H
Hosaka, T
Kawase, Y
Yasuda, K
Kikkawa, K
Yamauchi-Kohno, R
Yamada, K
JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (21) : 3369 - 3377
[24] Nicotinamide derivatives as a new class of gastric (H+/K+)-ATPase inhibitors .3. Synthesis and gastric antisecretory activity of 2-[(2- and 4-aminobenzyl, and alpha-methyllbenzyl)sulfinyl]-N-(4-pyridinyl)-3-pyridinecarboxamides
Terauchi, H
Tanitame, A
Tada, K
Nakamura, K
Seto, Y
Nishikawa, Y
CHEMICAL & PHARMACEUTICAL BULLETIN, 1997, 45 (07) : 1177 - 1182
[25] Synthesis and antiinflammatory activity of, 2-[5′-(4-pyridinyl)-1′,2′,3′-oxadiazol-2-yl-thiomethyl]-3-substituted-aryl-6-substituted-quinazolin-4-ones
Rajput, Chatrasal Singh
Kumar, Ashok
Bhati, Sudhir Kumar
Singh, Jai
ASIAN JOURNAL OF CHEMISTRY, 2008, 20 (08) : 6246 - 6252
[26] Potent and selective ET-A antagonists.: 1.: Syntheses and structure-activity relationships of N-(6-(2-(aryloxy)ethoxy)-4-pyrimidinyl)sulfonamide derivatives
Morimoto, H
Shimadzu, H
Kushiyama, E
Kawanishi, H
Hosaka, T
Kawase, Y
Yasuda, K
Kikkawa, K
Yamauchi-Kohno, R
Yamada, K
JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (21) : 3355 - 3368
[27] PYROPHTHALONES .7. SYNTHESIS AND ANTIINFLAMMATORY ACTIVITY OF 2-(4-PYRIDINYL)INDANE-1,3-DIONES DIVERSELY SUBSTITUTED ON THE BENZENE-RING
LEBLOIS, D
PIESSARD, S
LEBAUT, G
KUMAR, P
BRION, JD
SPARFEL, L
SANCHEZ, RY
JUGE, M
PETIT, JY
WELIN, L
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1987, 22 (03) : 229 - 238
[28] Nicotinamide derivatives as a new class of gastric (H+/K+)-ATPase inhibitors .2. Synthesis and structure-activity relationships of 2-[(2,4-dimethoxybenzyl)sulfinyl]-N-(4-pyridinyl)pyridine-3-carboxamides
Terauchi, H
Tanitame, A
Tada, K
Nakamura, K
Seto, Y
Nishikawa, Y
CHEMICAL & PHARMACEUTICAL BULLETIN, 1997, 45 (06) : 1027 - 1038
[29] AS601245 (1,3-benzothiazol-2-yl(2-{[2-(3-pyridinyl)ethyl]amino}-4 pyrimidinyl) acetonitrile):: A c-Jun NH2-terminal protein kinase inhibitor with neuroprotective properties
Carboni, S
Hiver, A
Szyndralewiez, C
Gaillard, P
Gotteland, JP
Vitte, PA
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2004, 310 (01): : 25 - 32
[30] Synthesis and dimeric crystal structure of sulfonylurea compound N-[2-(4-methyl)pyrimidinyl]-N′-2-methoxycarbonyl-benzene sulfonylurea
Wang, BL
Ning, M
Wang, JG
Ma, Y
Li, ZM
Leng, XB
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2004, 23 (07) : 783 - 787

← 1 2 3 4 5 →