IDENTIFICATION OF HUMAN LIVER CYTOCHROME P450S INVOLVED IN THE MICROSOMAL METABOLISM OF THE ANTIHISTAMINIC DRUG LORATADINE

被引:24
|
作者
YUMIBE, N [1 ]
HUIE, K [1 ]
CHEN, KJ [1 ]
CLEMENT, RP [1 ]
CAYEN, MN [1 ]
机构
[1] SCHERING PLOUGH CORP,RES INST,DEPT DRUG METAB & PHARMACOKINET,LAFAYETTE,NJ 07848
关键词
CYTOCHROME P450; METABOLISM; LORATADINE; DESCARBOETHOXYLORATADINE; KETOCONAZOLE; TROLEANDOMYCIN; QUINIDINE;
D O I
10.1159/000237063
中图分类号
R392 [医学免疫学];
学科分类号
100102 ;
摘要
[No abstract available]
引用
收藏
页码:420 / 420
页数:1
相关论文
共 50 条
  • [31] Identification of cytochrome P450s in human glioma cell line
    Vasquez, HG
    Strobel, H
    INTERNATIONAL JOURNAL OF ONCOLOGY, 1998, 12 (06) : 1291 - 1294
  • [32] Microsomal ethanol oxidizing system activity by human hepatic cytochrome P450s
    Asai, H
    Imaoka, S
    Kuroki, T
    Monna, T
    Funae, Y
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1996, 277 (02): : 1004 - 1009
  • [33] Functioning of Microsomal Cytochrome P450s: Murbum Concept Explains the Metabolism of Xenobiotics in Hepatocytes
    Manoj, Kelath Murali
    Parashar, Abhinav
    Gade, Sudeep K.
    Venkatachalam, Avanthika
    FRONTIERS IN PHARMACOLOGY, 2016, 7
  • [34] Effects of ginsenosides on the expression of cytochrome P450s and transporters involved in cholesterol metabolism
    Kawase, Atsushi
    Yamada, Ayano
    Gamou, Yuko
    Tahara, Chika
    Takeshita, Fumiaki
    Murata, Kazuya
    Matsuda, Hideaki
    Samukawa, Keiichi
    Iwaki, Masahiro
    JOURNAL OF NATURAL MEDICINES, 2014, 68 (02) : 395 - 401
  • [35] Identification of human liver cytochrome P450 isoforms involved in the in vitro metabolism of cyclobenzaprine
    Wang, RW
    Liu, LD
    Cheng, HY
    DRUG METABOLISM AND DISPOSITION, 1996, 24 (07) : 786 - 791
  • [36] Identification of cytochrome P450 isoforms involved in the metabolism of loperamide in human liver microsomes
    Kyoung-Ah Kim
    Jaegul Chung
    Dong-Hae Jung
    Ji-Young Park
    European Journal of Clinical Pharmacology, 2004, 60 : 575 - 581
  • [37] Identification of cytochrome P450 isoforms involved in the metabolism of loperamide in human liver microsomes
    Kim, KA
    Chung, JG
    Jung, DH
    Park, JY
    EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 2004, 60 (08) : 575 - 581
  • [38] An Unprecedented Number of Cytochrome P450s Are Involved in Secondary Metabolism in Salinispora Species
    Malinga, Nsikelelo Allison
    Nzuza, Nomfundo
    Padayachee, Tiara
    Syed, Puleng Rosinah
    Karpoormath, Rajshekhar
    Gront, Dominik
    Nelson, David R.
    Syed, Khajamohiddin
    MICROORGANISMS, 2022, 10 (05)
  • [39] Effects of ginsenosides on the expression of cytochrome P450s and transporters involved in cholesterol metabolism
    Atsushi Kawase
    Ayano Yamada
    Yuko Gamou
    Chika Tahara
    Fumiaki Takeshita
    Kazuya Murata
    Hideaki Matsuda
    Keiichi Samukawa
    Masahiro Iwaki
    Journal of Natural Medicines, 2014, 68 : 395 - 401
  • [40] Identification of cytochromes P450 involved in human liver microsomal metabolism of ecabapide, a prokinetic agent
    Fujimaki, Y
    Arai, N
    Inaba, T
    XENOBIOTICA, 1999, 29 (12) : 1273 - 1282