IRREVERSIBLE BLOCKADE OF NICOTINIC ACETYLCHOLINE-RECEPTOR AGONIST ANTAGONIST SITES BY LOPHOTOXIN

被引:0
|
作者
CULVER, P [1 ]
TAYLOR, P [1 ]
机构
[1] UNIV CALIF SAN DIEGO,DIV PHARMACOL,LA JOLLA,CA 92093
关键词
D O I
暂无
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:1144 / 1144
页数:1
相关论文
共 50 条
  • [41] STRUCTURE, OLIGOSACCHARIDE STRUCTURES, AND POSTTRANSLATIONALLY MODIFIED SITES OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    POULTER, L
    EARNEST, JP
    STROUD, RM
    BURLINGAME, AL
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1989, 86 (17) : 6645 - 6649
  • [42] BINDING OF DEPOLARIZING DRUGS TO THE IONIC CHANNEL SITES OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    ELDEFRAWI, AT
    MILLER, ER
    ELDEFRAWI, ME
    BIOCHEMICAL PHARMACOLOGY, 1982, 31 (09) : 1819 - 1822
  • [43] DETERMINATION OF THE SITES OF CAMP-DEPENDENT PHOSPHORYLATION ON THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    YEE, GH
    HUGANIR, RL
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1987, 262 (34) : 16748 - 16753
  • [44] ANTIGENIC SITES OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR CHARACTERIZED BY STABILITY TO ACID DENATURATION
    BARKAS, T
    JAMES, RW
    EDER, L
    FULPIUS, BW
    BIOCHEMICAL SOCIETY TRANSACTIONS, 1984, 12 (05) : 814 - 815
  • [45] NICOTINIC ACETYLCHOLINE-RECEPTOR ION CHANNEL BLOCKADE BY COCAINE - THE MECHANISM OF SYNAPTIC ACTION
    SWANSON, KL
    ALBUQUERQUE, EX
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1987, 243 (03): : 1202 - 1210
  • [46] GANGLIONIC NICOTINIC ACETYLCHOLINE-RECEPTOR ACTIVATION BY THE NOVEL AGONIST ABT-418
    BRIGGS, CA
    HUGHES, ML
    MONTEGGIA, LM
    GIORDANO, T
    DONNELLYROBERTS, D
    ARNERIC, SP
    DRUG DEVELOPMENT RESEARCH, 1995, 34 (01) : 39 - 46
  • [47] THE INFLUENCE OF ANTIBIOTICS ON AGONIST OCCUPATION AND FUNCTIONAL-STATES OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    BROWN, RD
    TAYLOR, P
    MOLECULAR PHARMACOLOGY, 1983, 23 (01) : 8 - 16
  • [48] THE NARCOTIC-ANTAGONIST NALTREXONE HAS A BIPHASIC EFFECT ON THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    MADSEN, BW
    ALBUQUERQUE, EX
    FEBS LETTERS, 1985, 182 (01): : 20 - 24
  • [49] THE REACTION SITE OF A NONCOMPETITIVE ANTAGONIST IN THE DELTA-SUBUNIT OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    OBERTHUR, W
    MUHN, P
    BAUMANN, H
    LOTTSPEICH, F
    WITTMANNLIEBOLD, B
    HUCHO, F
    EMBO JOURNAL, 1986, 5 (08): : 1815 - 1819
  • [50] FUNCTIONAL DOMAINS OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    WEISE, C
    MACHOLD, J
    KREIENKAMP, HJ
    TSETLIN, V
    UTKIN, Y
    HUCHO, F
    BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1991, 372 (10): : 911 - 912