SYNTHESIS OF FUNCTIONALIZED INDOLES BY DIELS-ALDER REACTION UTILIZING THE DIENE GENERATED BY THE ALKYLATION OF N-METHYL-3-THIOACETYLPYRROLE

被引：0
|
作者：
MURASE, M [1 ]
YOSHIDA, S [1 ]
HOSAKA, T [1 ]
TOBINAGA, S [1 ]
机构：
[1] SHOWA COLL PHARMACEUT SCI, TOKYO 194, JAPAN
来源：
CHEMICAL & PHARMACEUTICAL BULLETIN | 1991年 / 39卷 / 02期
关键词：
CYCLOADDITION; 3-VINYLPYRROLE; 1-METHYL-3-THIOACETYLPYRROLE; ALKYLATION; DIENOPHILE; INDOLE;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
Cycloaddition reaction of 3-vinylpyrroles, generated by the alkylation of 1-methyl-3-thioacetylpyrrole, with dienophiles provided functionalized indoles.
引用
收藏
页码：489 / 492
页数：4
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