Kinetics and mechanism of inhibition of serine esterases by fluorinated carbethoxy 1-aminophosphonates

被引:0
|
作者
G. F. Makhaeva
S. V. Lushchekina
O. G. Serebryakova
A. Yu. Aksinenko
T. V. Goreva
R. J. Richardson
I. V. Martynov
机构
[1] Russian Academy of Sciences,Institute of Physiologically Active Compounds
[2] Russian Academy of Sciences,Emanuel Institute of Biochemical Physics
[3] University of Michigan,Department of Environmental Health Sciences
来源
关键词
DOKLADY Biochemistry; Serine Hydrolase; Electron Acceptor Substituent; Butyrylthio Choline; Serine Esterase;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:203 / 206
页数:3
相关论文
共 19 条
  • [1] Kinetics and mechanism of inhibition of serine esterases by fluorinated carbethoxy 1-aminophosphonates
    Makhaeva, G. F.
    Lushchekina, S. V.
    Serebryakova, O. G.
    Aksinenko, A. Yu.
    Goreva, T. V.
    Richardson, R. J.
    Martynov, I. V.
    DOKLADY BIOCHEMISTRY AND BIOPHYSICS, 2013, 451 (01) : 203 - 206
  • [2] Kinetics and mechanism of inhibition of serine esterases by fluorinated aminophosphonates
    Makhaeva, G. F.
    Aksinenko, A. Y.
    Sokolov, V. B.
    Baskin, I. I.
    Palyulin, V. A.
    Zefirov, N. S.
    Hein, N. D.
    Kampf, J. W.
    Wijeyesakere, S. J.
    Richardson, R. J.
    CHEMICO-BIOLOGICAL INTERACTIONS, 2010, 187 (1-3) : 177 - 184
  • [3] Kinetics and Mechanism of Inhibition of a Serine β-Lactamase by O-Aryloxycarbonyl Hydroxamates
    Pelto, Ryan B.
    Pratt, R. F.
    BIOCHEMISTRY, 2008, 47 (46) : 12037 - 12046
  • [4] MECHANISM OF END PRODUCT INHIBITION OF SERINE BIOSYNTHESIS .I. PURIFICATION AND KINETICS OF PHOSPHOGLYCERATE DEHYDROGENASE
    SUGIMOTO, E
    PIZER, LI
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1968, 243 (09) : 2081 - &
  • [5] Mechanism of differential inhibition of hepatic and pancreatic fatty acid ethyl ester synthase by inhibitors of serine-esterases: in vitro and cell culture studies
    Kaphalia, BS
    Mericle, KA
    Ansari, GAS
    TOXICOLOGY AND APPLIED PHARMACOLOGY, 2004, 200 (01) : 7 - 15
  • [6] The mechanism of inhibition of antibody-based inhibitors of membrane-type serine protease 1 (MT-SP1)
    Farady, Christopher J.
    Sun, Jeonghoon
    Darragh, Molly R.
    Miller, Susan M.
    Craik, Charles S.
    JOURNAL OF MOLECULAR BIOLOGY, 2007, 369 (04) : 1041 - 1051
  • [7] Insight into the Dual Inhibition Mechanism of Corilagin against MRSA Serine/Threonine Phosphatase (Stp1) by Molecular Modeling
    Yang, Yanan
    Wang, Xiyan
    Gao, Yawen
    Niu, Xiaodi
    ACS OMEGA, 2020, 5 (51): : 32959 - 32968
  • [8] Pim-1 ligand-bound structures reveal the mechanism of serine/threonine kinase inhibition by LY294002
    Jacobs, MD
    Black, J
    Futer, O
    Swenson, L
    Hare, B
    Fleming, M
    Saxena, K
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2005, 280 (14) : 13728 - 13734
  • [9] ENZYME-KINETICS OF LACTATE-DEHYDROGENASE ISOENZYMES AND THE MECHANISM OF CHEMICAL INHIBITION FOR THE BMD LD-1 ASSAY
    ONIGBINDE, TA
    WU, AHB
    WU, YS
    SIMMONS, MJ
    CLINICAL CHEMISTRY, 1990, 36 (06) : 1135 - 1135
  • [10] Structural Bases for Hesperetin Derivatives: Inhibition of Protein Tyrosine Phosphatase 1B, Kinetics Mechanism and Molecular Docking Study
    Ali, Md Yousof
    Jannat, Susoma
    Jung, Hyun-Ah
    Choi, Jae-Sue
    MOLECULES, 2021, 26 (24):