[18F]F15599, a novel 5-HT1A receptor agonist, as a radioligand for PET neuroimaging

被引：0
|
作者：
Laëtitia Lemoine
Mathieu Verdurand
Bernard Vacher
Elodie Blanc
Didier Le Bars
Adrian Newman-Tancredi
Luc Zimmer
机构：
[1] Université de Lyon,Laboratory of Neuropharmacology
[2] CERMEP – Imagerie du Vivant,PET Department
[3] CERMEP – Imagerie du Vivant,ANIMAGE Department
[4] Centre de Recherches Pierre Fabre,undefined
来源：
European Journal of Nuclear Medicine and Molecular Imaging | 2010年 / 37卷
关键词：
Serotonin 1A receptor; PET; Agonist; Rat; Cat;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：594 / 605
页数：11
相关论文
共 50 条
  • [21] EVALUATION OF [18F]FPWAY AND [18F]FBWAY, 5-HT1A RECEPTOR PET LIGANDS, FOR SENSITIVITY TO ENDOGENOUS 5-HT IN RAT
    Jagoda, E. M.
    Lang, L.
    Tokugawa, J.
    Ma, Y.
    Contoreggi, C.
    Eckelman, W. C.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2005, 48 : S74 - S74
  • [22] Evaluation of [18F]SL702 as a prospective agonist PET radioligand for brain 5-HT1A receptors in mice and monkey
    Lu, Shuiyu
    Liow, J. S.
    Zoghbi, S. S.
    Gladding, R. L.
    Innis, R. B.
    Pike, V. W.
    NEUROIMAGE, 2008, 41 : T157 - T158
  • [23] Initial evaluation of [18F]F13714, a novel 5-HT1A receptor agonist in non-human primates
    Tavares, A.
    Becker, G.
    Barret, O.
    Morley, T.
    Alagille, D.
    Vacher, B.
    Newman-Tancredi, A.
    Tamagnan, G.
    Zimmer, L.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2013, 40 : S144 - S144
  • [24] Antidepressant- and anxiolytic-like effects of "biased'' 5-HT1A receptor agonists F15599 and F13714 in rats
    Jastrzebska-Wiesek, Magdalena
    Partyka, Anna
    Wasik, Anna
    Sniecikowska, Joanna
    Newman-Tancredi, Adrian
    Wesolowska, Anna
    PHARMACOLOGICAL REPORTS, 2015, 67 : 23 - 23
  • [25] [18F]F13640: a selective agonist PET radiopharmaceutical for imaging functional 5-HT1A receptors in humans
    Courault, Pierre
    Lancelot, Sophie
    Costes, Nicolas
    Colom, Matthieu
    Le Bars, Didier
    Redoute, Jerome
    Gobert, Florent
    Dailler, Frederic
    Isal, Sibel
    Iecker, Thibaut
    Newman-Tancredi, Adrian
    Merida, Ines
    Zimmer, Luc
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2023, 50 (06) : 1651 - 1664
  • [26] [18F]F13640: a selective agonist PET radiopharmaceutical for imaging functional 5-HT1A receptors in humans
    Pierre Courault
    Sophie Lancelot
    Nicolas Costes
    Matthieu Colom
    Didier Le Bars
    Jérôme Redoute
    Florent Gobert
    Frédéric Dailler
    Sibel Isal
    Thibaut Iecker
    Adrian Newman-Tancredi
    Inés Merida
    Luc Zimmer
    European Journal of Nuclear Medicine and Molecular Imaging, 2023, 50 : 1651 - 1664
  • [27] Synthesis and preliminary evaluation of [18F] S14506 as a novel PET radioligand for brain 5-HT1A receptors in rat
    Lu, S. Y.
    Liow, J. S.
    Zoghbi, S. S.
    Brown, A. K.
    Musachio, J. L.
    Vermeulen, E. S.
    Wikstrom, H. V.
    Innis, R. B.
    Pike, V. W.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2005, 32 : S52 - S52
  • [28] Aggression-reducing effects of F15599, a novel selective 5-HT1A receptor agonist, after microinjection into the ventral orbital prefrontal cortex, but not in infralimbic cortex in male mice
    Stein, Dirson Joao
    Miczek, Klaus A.
    Lucion, Aldo Bolten
    Martins de Almeida, Rosa Maria
    PSYCHOPHARMACOLOGY, 2013, 230 (03) : 375 - 387
  • [29] Development of an 18F-labelled 5-HT2A receptor agonist PET radioligand
    Ettrup, Anders
    Hansen, Martin
    Gillings, Nic
    Dyssegaard, Agnete
    Lehel, Szabolcs
    Hansen, Hanne D.
    Herth, Matthias M.
    Madsen, Jacob
    Kristensen, Jepser
    Knudsen, Gitte M.
    JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 2012, 32 : S109 - S109
  • [30] F15599, a highly selective post-synaptic 5-HT1A receptor agonist: in-vivo profile in behavioural models of antidepressant and serotonergic activity
    Assie, Marie-Bernadette
    Bardin, Laurent
    Auclair, Agnes L.
    Carilla-Durand, Elisabeth
    Depoortere, Ronan
    Koek, Wouter
    Kleven, Mark S.
    Colpaert, Francis
    Vacher, Bernard
    Newman-Tancredi, Adrian
    INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY, 2010, 13 (10): : 1285 - 1298
12345