Polyfunctional imidazoles: VIII. 1-Aryl-4-chloro-5-[R-sulfanyl(sulfonyl)methyl]-1H-imidazoles

被引：0
|
作者：
A. N. Grozav
V. A. Chornous
A. A. Palamar
M. V. Vovk
机构：
[1] Bukovinian State Medical University,Institute of Organic Chemistry
[2] National Academy of Sciences of Ukraine,undefined
来源：
Russian Journal of Organic Chemistry | 2014年 / 50卷
关键词：
Potassium Permanganate; Methanethiol; Chloroacetic Acid; Sulfanyl; Methylsulfanyl;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Alkylation of (1-aryl-4-chloro-1H-imidazol-5-yl)methanethiols with alkyl halides, propargyl bromide, or chloroacetic acid gave 1-aryl-5-(R-sulfanylmethyl)-4-chloro-1H-imidazoles. 1-Aryl-4-chloro-5-(methylsulfanylmethyl)-1H-imidazoles and [(1-aryl-4-chloro-1H-imidazol-5-yl)methylsulfanyl]acetic acids were oxidized to the corresponding sulfones with potassium permanganate.
引用
收藏
页码：1335 / 1340
页数：5
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