NMR-based platform for fragment-based lead discovery used in screening BRD4-targeted compounds

被引：0
|
作者：
Jun-lan Yu
Tian-tian Chen
Chen Zhou
Fu-lin Lian
Xu-long Tang
Yi Wen
Jing-kang Shen
Ye-chun Xu
Bing Xiong
Nai-xia Zhang
机构：
[1] Shanghai Institute of Materia Medica,Department of Analytical Chemistry
[2] Chinese Academy of Sciences,undefined
[3] China & University of Chinese Academy of Sciences,undefined
[4] CAS Key Laboratory of Receptor Research,undefined
[5] Drug Discovery and Design Center,undefined
[6] Shanghai Institute of Materia Medica,undefined
[7] Chinese Academy of Sciences,undefined
[8] State Key Laboratory of Drug Research,undefined
[9] Shanghai Institute of Materia Medica,undefined
[10] Chinese Academy of Sciences,undefined
来源：
Acta Pharmacologica Sinica | 2016年 / 37卷
关键词：
fragment-based lead discovery; NMR; bromodomain; BRD4 inhibitors;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：984 / 993
页数：9
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