Radiosynthesis and evaluation of [18F]FMTP, a COX-2 PET ligand

被引：0
|
作者：
J. S. Dileep Kumar
Jaya Prabhakaran
Andrei Molotkov
Anirudh Sattiraju
Jongho Kim
Mikhail Doubrovin
J. John Mann
Akiva Mintz
机构：
[1] New York State Psychiatric Institute,Molecular Imaging and Neuropathology Division
[2] Columbia University Medical Center,Department of Psychiatry
[3] Columbia University Medical Center,Department of Radiology
来源：
Pharmacological Reports | 2020年 / 72卷
关键词：
PET; COX-2; Radiotracer; Inflammation; Brain;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
引用
收藏
页码：1433 / 1440
页数：7
相关论文
共 50 条
  • [11] Re(CO)3([18F]FEDA), a novel 18F PET renal tracer: Radiosynthesis and preclinical evaluation
    Lipowska, Malgorzata
    Jarkas, Nashwa
    Voll, Ronald J.
    Nye, Jonathon A.
    Klenc, Jeffrey
    Goodman, Mark M.
    Taylor, Andrew T.
    NUCLEAR MEDICINE AND BIOLOGY, 2018, 58 : 42 - 50
  • [12] Synthesis and evaluation of ortho-[18F]fluorocelecoxib for COX-2 cholangiocarcinoma imaging
    Chang, Chi-Wei
    Yeh, Chun-Nan
    Chung, Yi-Hsiu
    Chen, Yong-Ren
    Tien, Shi-Wei
    Chen, Tsung-Wen
    Farn, Shiou-Shiow
    Huang, Ying-Cheng
    Yu, Chung-Shan
    DRUG DESIGN DEVELOPMENT AND THERAPY, 2018, 12 : 1467 - 1478
  • [13] Characterization of the radiosynthesis and purification of [18F]THK-5351, a PET ligand for neurofibrillary tau
    Betthauser, Tobey J.
    Ellison, Paul A.
    Murali, Dhanabalan
    Lao, Patrick J.
    Barnhart, Todd E.
    Furtunoto, Shozo
    Okamura, Nobuyuki
    Johnson, Sterling C.
    Engle, Jonathan W.
    Nickles, Robert J.
    Christian, Bradley T.
    APPLIED RADIATION AND ISOTOPES, 2017, 130 : 230 - 237
  • [14] Radiosynthesis, in vitro and preliminary in vivo evaluation of the novel glutamine derived PET tracers [18F]fluorophenylglutamine and [18F] fluorobiphenylglutamine
    Baguet, Tristan
    Verhoeven, Jeroen
    Pauwelyn, Glenn
    Hu, Jiyun
    Lambe, Patricia
    De Lombaerde, Stef
    Piron, Sarah
    Donche, Sam
    Descamps, Benedicte
    Goethals, Ingeborg
    Vanhove, Christian
    De Vos, Filip
    Beyzavi, M. Hassan
    NUCLEAR MEDICINE AND BIOLOGY, 2020, 86-87 : 20 - 29
  • [15] SYNTHESIS OF 18F RADIOLABELED COX189, A SELECTIVE COX-2 INHIBITOR
    Murali, D.
    Bordeaux, K.
    Ray, T.
    Ciszewska, G.
    Tse, F.
    Nickles, R. J.
    Dejesus, O. T.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2009, 52 : S152 - S152
  • [16] Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors
    Wilson, Alan A.
    Garcia, Armando
    Parkes, Jun
    McCormick, Patrick
    Stephenson, Karin A.
    Houle, Sylvain
    Vasdev, Neil
    NUCLEAR MEDICINE AND BIOLOGY, 2008, 35 (03) : 305 - 314
  • [17] Radiosynthesis and evaluation of novel 18F labeled PET ligands for imaging monoacylglycerol lipase
    Li, Yinlong
    Mori, Wakana
    Chaudhary, Ahmad
    Zhao, Chunyu
    Yamasaki, Tomoteru
    Zhang, Zachary
    Feng, Siyan
    Ware, Tim
    Rong, Jian
    Fujinaga, Masayuki
    Chen, Jiahui
    Kumata, Katsushi
    Zhang, Yiding
    Hu, Kuan
    Xie, Lin
    Zhou, Xin
    Song, Zhendong
    Gao, Yabiao
    Sun, Zhenkun
    Patel, Jimmy S.
    Zhai, Chuangyan
    Yuan, Katherine Y.
    Collier, Thomas L.
    Ran, Chongzhao
    Collin, Ludovic
    Haider, Achi
    Grether, Uwe
    Wittwer, Matthias B.
    Cravatt, Benjamin F.
    Zhang, Ming-Rong
    Liang, Steven H.
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 285
  • [18] Radiosynthesis and evaluation of [18F]AFM, a selective PET tracer for the serotonin transporter.
    Huang, Y
    Bac, SA
    Zhu, Z
    Hwang, DR
    Narendran, R
    Talbot, PS
    Hackett, E
    Kegeles, LS
    Laruelle, M
    JOURNAL OF NUCLEAR MEDICINE, 2002, 43 (05) : 358P - 358P
  • [19] FLUO 14-Synthesis and in vivo evaluation of [18F]labeled COX-2 inhibitors
    Kumar, J. S. Dileep
    Mann, J. John
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 960 - 960
  • [20] Automated Radiosynthesis and Biological Evaluation of [18F]FSPG
    Glaser, Matthias
    Gendron, Thibault
    McCormick, Patrick
    Berndt, Mathias
    Koglin, Norman
    Sander, Kerstin
    Witney, Tim
    Arstad, Erik
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2017, 60 : S171 - S171
12345