Synthesis, characterization, antibacterial and antifungal activity of thienopyrimidines and triazolothienopyrimidines

被引：0
|
作者：
S. I. Panchamukhi
A. K. Mohammed Iqbal
A. Y. Khan
M. B. Kalashetti
I. M. Khazi
机构：
[1] Karnatak University,Department of Chemistry
来源：
Pharmaceutical Chemistry Journal | 2011年 / 44卷
关键词：
Triazolothienopyrimidines; Gewald reaction; antibacterial activity; antifungal activity;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Aseries of novel triazole fused tetracyclic thienopyrimidines (III – X) were synthesized from the corresponding precursor 5-amino-4-cyano-3-methylthiophene-2-carboxylic acid ethyl ester I. The precursor were in turn prepared via the Gewald reaction. Structures of all the newly synthesized compounds were characterized by spectral and analytical data. All the tested compounds displayed promising antibacterial and antifungal activities.
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页码：694 / 696
页数：2
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