Reactivity study of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione toward the synthesis of bicyclic 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione analogues

被引：15

作者：

Brouillette, Yann ^{[1
]}

Lisowski, Vincent ^{[1
]}

Fulcrand, Pierre ^{[1
]}

Martinez, Jean ^{[1
]}

机构：

[1] Univ Montpellier 2, UFR Sci Pharmaceut & Biol, CNRS, UMR 5810,LAPP, F-34093 Montpellier 5, France

来源：

JOURNAL OF ORGANIC CHEMISTRY | 2007年 / 72卷 / 07期

关键词：

EFFICIENT SYNTHESIS; RING; ANTAGONISTS; PREDICTION; DISCOVERY; KINETICS; XANTHINE; AGENTS;

D O I：

10.1021/jo0622882

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[GRAPHIC] A series of 10 optically pure 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione derivatives has been synthesized in 41-75% yields on treatment of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione with different natural alpha-amino acids.

引用

页码：2662 / 2665

页数：4

共 50 条

[41] SYNTHESIS AND CHEMISTRY OF SOME THIENO[3,2-D]-1,2,3-TRIAZIN-4(3H)-ONES
HUDDLESTON, PR
BARKER, JM
ADAMCZEWSKA, YZ
WOOD, ML
HOLMES, D
JOURNAL OF CHEMICAL RESEARCH-S, 1993, (02): : 72 - 73
[42] SYNTHESIS OF 4,5-DIHYDRO-1H,3H-THIENO[3,4-C]THIOPHENE AND 4,5-DIHYDRO-1H,3H-THIENO[3,4-C]FURAN
RIPOLL, JL
VALLEE, Y
KHALID, M
HAKIKI, A
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1992, 29 (07) : 1867 - 1868
[43] 2H,10H-1,4-dioxepino[5′,6′:4,5]thieno[3,2-e][1,4]dioxepine-5,7(3H,9H)-dione
Tomura, Masaaki
Ono, Katsuhiko
Kaiden, Masanori
Tsukamoto, Kenichi
Saito, Katsuhiro
ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2007, 63 : O4568 - U3757
[44] A FACILE SYNTHESIS AND DOCKING STUDIES OF PYRIDINE CONTAINING 1H-THIENO[3,2-C]PYRAZOLE
Madipelly, Rajeshwari
HETEROCYCLIC LETTERS, 2020, 10 (03): : 509 - 515
[45] Facile synthesis of 2-(substituted amino)-4H-thieno[3,2-e]-1,3-thiazin-4-ones
Rajab Abu-El-Halawa
Alaa Sarabi
Mustafa M. El-Abadelah
Monatshefte für Chemie - Chemical Monthly, 2008, 139
[46] Synthesis of a new pyrrolo[1,3]diazepine: 4H-pyrrolo[1,2-a]thieno[2,3-e][1,3]diazepine
Daich, A
Ohier, P
Decroix, B
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1995, 32 (06) : 1731 - 1734
[47] PYRROLOPYRIMIDINES .1. ELECTROPHILIC SUBSTITUTION-REACTIONS OF 1,3-DIMETHYLPYRROLO[3,2-D]PYRIMIDINE-2,4-DIONE
TSUPAK, EB
TKACHENKO, YN
POZHARSKY, AF
KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 1994, (09): : 1242 - 1248
[48] INTRAMOLECULAR CYCLIZATION - SYNTHESIS OF 9-OXO-4H,9H-PYRROLO[1,2-A]THIENO[2,3-D]PYRIDINE AND 4-OXO-4H,9H-PYRROLO[1,2-A]THIENO[2,3-D]PYRIDINE - SYNTHESIS OF PYRROLO[1,2-A]THIENO[3,2-E][1,4]DIAZEPINE AND PYRROLO[1,2-A]THIENO[2,3-E][1,4]DIAZEPINE
DECROIX, B
MOREL, J
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1991, 28 (01) : 81 - 87
[49] SYNTHESIS OF 4-H-AMINO-6 PYRROLO [1,2-A] THIENO [3,2-F] DIAZEPINE-1,4
RAULT, S
CUGNONDESEVRICOURT, M
ELKHASHEF, H
ROBBA, M
COMPTES RENDUS HEBDOMADAIRES DES SEANCES DE L ACADEMIE DES SCIENCES SERIE C, 1980, 290 (09): : 169 - 171
[50] Pyrrolopyrimidines.: 3.: 5-amino-1,3-dimethylpyrrolo[3,2-d]pyrimidine-2,4(1H,3H)-dione
Tkachenko, YN
Tsupak, EB
Pozharsky, AF
KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII, 1999, (03): : 375 - 380

← 1 2 3 4 5 →