SYNTHESIS OF NEWER STEROIDAL PYRAZOLES AS PROSPECTIVE ANTIMICROBIAL AND ANTIINFLAMMATORY AGENTS

被引：0

作者：

Murti, Y. ^{[1
]}

Sharma, A. ^{[1
]}

Pathak, D. ^{[1
]}

机构：

[1] Rajiv Acad Pharm, Dept Pharmaceut Chem, Mathura 281001, India

来源：

INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2009年 / 19卷 / 02期

关键词：

BIOLOGICAL-ACTIVITY;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of newer steroidal pyrazoles (C(1)-C(4)) have been synthesized by the reaction of 3-chloro-cholest-2,4-dien-2-aldehyde with hydrazine hydrate, phenyl hydrazine, p-fluorophenyl hydrazine and 2,4-dinitrophenyl hydrazine respectively. The constitutions of all the compounds have been established by elemental analyses, FTIR and (1)H NMR spectral data. All the compounds were screened for their antimicrobial and antiinflammatory activity under identical conditions.

引用

页码：183 / 184

页数：2

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