The objective was to investigate the effects of heat pretreatment and simulated gastrointestinal digestion on potential antioxidant, anticancer and anti-inflammatory activities of hempseed (Cannabis sativa L.) proteins. Unheated isolated hempseed protein (IHP) and its heated counterparts (100 degrees C, 15 min and 30 min, termed as HP15D and HP30D) were hydrolyzed sequentially with pepsin and pancreatin and analyzed for digestibility and bioactivity (antioxidant, anti-proliferative and anti-inflammatory properties). Heat pretreatment led to an increase of low molecular weight proteins and degree of hydrolysis, and decrease of concentration of soluble protein, which means heat pretreated can significantly improve the digestibility of IHP. Pepsin-pancreatin digests released from heat pretreated IHP possessed less antioxidant, antiproliferative and anti-inflammatory properties than digests from unheated IHP. In conclusion, heat pre-treatment improved the digestibility of IHP but the resulting digests from heated IHP had lower bioactivity.
机构:
Univ Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Univ Autonoma Estado Hidalgo, Area Acad Quim, Mineral De La Reforma, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Baruchs Munoz-Llandes, Ciro
Araceli Guzman-Ortiz, Fabiola
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Univ Autonoma Estado Hidalgo, Area Acad Quim, Mineral De La Reforma, Hidalgo, Mexico
Univ Autonoma Estado Hidalgo, CONACYT, Mineral De La Reform, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Araceli Guzman-Ortiz, Fabiola
Delia Roman-Gutierrez, Alma
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Univ Autonoma Estado Hidalgo, Area Acad Quim, Mineral De La Reforma, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Delia Roman-Gutierrez, Alma
Maria Palma-Rodriguez, Heidi
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Univ Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Maria Palma-Rodriguez, Heidi
Castro-Rosas, Javier
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Univ Autonoma Estado Hidalgo, Area Acad Quim, Mineral De La Reforma, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Castro-Rosas, Javier
Hernandez-Sanchez, Humberto
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Inst Politecn Natl, Dept Ingn Bioquim, Escuela Nacl Ciencias Biol, Unidad Zacatenco, Ciudad De Mexico, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Hernandez-Sanchez, Humberto
Francisco Zamora-Natera, Juan
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Univ Guadalajara, Ctr Univ Ciencias Biol & Agr, Dept Bot & Zool, Zapopan, Jalisco, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
Francisco Zamora-Natera, Juan
Vargas-Torres, Apolonio
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Univ Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, MexicoUniv Autonoma Estado Hidalgo, Rancho Univ, Inst Ciencias Agr, Tulancingo De Bravo, Hidalgo, Mexico
机构:
Univ Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Univ Rhode Isl, George & Anne Ryan Inst Neurosci, Kingston, RI 02881 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Puopolo, Tess
Chang, Tanran
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Chinese Acad Sci, Inst Proc Engn, State Key Lab Biochem Engn, Beijing 100190, Peoples R China
Univ Chinese Acad Sci, Beijing 100049, Peoples R ChinaUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Chang, Tanran
Liu, Chang
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Univ Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Liu, Chang
Li, Huifang
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Univ Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Li, Huifang
Liu, Xu
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Yunnan Hempmon Pharmaceut Co Ltd, Kunming 650032, Yunnan, Peoples R ChinaUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Liu, Xu
Wu, Xian
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Miami Univ, Dept Kinesiol Nutr & Hlth, Oxford, OH 45056 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Wu, Xian
Ma, Hang
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Univ Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Univ Rhode Isl, George & Anne Ryan Inst Neurosci, Kingston, RI 02881 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Ma, Hang
Seeram, Navindra P.
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机构:
Univ Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA
Univ Rhode Isl, George & Anne Ryan Inst Neurosci, Kingston, RI 02881 USAUniv Rhode Isl, Coll Pharm, Dept Biomed & Pharmaceut Sci, Bioact Bot Res Lab, Kingston, RI 02881 USA