Fragment-based approaches to type 2 kinase inhibitors

被引：0
|
作者：
Johnson, Christopher [1 ]
机构：
[1] Astex Pharmaceut, Cambridge, England
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2016年 / 251卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
239
引用
收藏
页数：1
相关论文
共 50 条
  • [31] Fragment-based design of SARS-CoV-2 Mpro inhibitors
    Teli, Divya M.
    Patel, Bansari
    Chhabria, Mahesh T.
    STRUCTURAL CHEMISTRY, 2022, 33 (06) : 2155 - 2168
  • [32] Fragment-based discovery of potent ERK2 pyrrolopyrazine inhibitors
    Burdick, Daniel J.
    Wang, Shumei
    Heise, Christopher
    Pan, Borlan
    Drummond, Jake
    Yin, JianPing
    Goeser, Lauren
    Magnuson, Steven
    Blaney, Jeff
    Moffat, John
    Wang, Weiru
    Chen, Huifen
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (21) : 4728 - 4732
  • [33] Computational fragment-based design of Wee1 kinase inhibitors with tricyclic core scaffolds
    Abdullah, Maaged
    Guruprasad, Lalitha
    STRUCTURAL CHEMISTRY, 2019, 30 (01) : 213 - 226
  • [34] Computational fragment-based design of Wee1 kinase inhibitors with tricyclic core scaffolds
    Maaged Abdullah
    Lalitha Guruprasad
    Structural Chemistry, 2019, 30 : 213 - 226
  • [35] Fragment-based Discovery of S100B Inhibitors Combining Computational and Biophysical Approaches
    Mangani, Stefano
    Cesari, Lucia
    Andreini, Matteo
    Lalli, Daniela
    del Conte, Rebecca
    Turano, Paola
    Padova, Alessandro
    Agamennone, Mariangela
    ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES, 2009, 65 : S302 - S303
  • [36] Drugging challenging targets using fragment-based approaches
    Coyne, Anthony G.
    Scott, Duncan E.
    Abell, Chris
    CURRENT OPINION IN CHEMICAL BIOLOGY, 2010, 14 (03) : 299 - 307
  • [37] Fragment-based discovery of the first known inhibitors of PHGDH
    Fuller, Nathan
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250
  • [38] Fragment-Based Deconstruction of Bcl-xL Inhibitors
    Barelier, Sarah
    Pons, Julien
    Marcillat, Olivier
    Lancelin, Jean-Marc
    Krimm, Isabelle
    JOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (06) : 2577 - 2588
  • [39] Fragment-based approach to covalent inhibitors of catalytic cysteines
    Kathman, Stefan
    Xu, Ziyang
    Statsyuk, Alexander
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 246
  • [40] Fragment-Based Screening for Enzyme Inhibitors Using Calorimetry
    Recht, Michael I.
    Nienaber, Vicki
    Torres, Francisco E.
    CALORIMETRY, 2016, 567 : 47 - 69
12345